| Nome |
# |
|
Cyclic RGD peptidomimetics containing bifunctional diketopiperazine scaffolds as new potent integrin ligands, file e2188be6-0032-4564-e053-6605fe0a49d6
|
561
|
|
Stereocontrolled Synthesis of Polyketide Libraries - Boron-Mediated Aldol Reactions with Aldehydes on Solid Support., file e2188be5-f7e2-4564-e053-6605fe0a49d6
|
487
|
|
Toward the First Nonpeptidic Molecular Tong Inhibitor of Wild-Type and Mutated HIV-1 Protease Dimerization, file e2188be5-fe24-4564-e053-6605fe0a49d6
|
350
|
|
Rhodium-catalyzed asymmetric hydrogenation of olefins with PhthalaPhos, a new class of chiral supramolecular ligands, file e2188be6-0031-4564-e053-6605fe0a49d6
|
326
|
|
Synthesis and Biological Evaluation (in Vitro and in Vivo) of Cyclic RGD Peptidomimetic - Paclitaxel Conjugates Targeting Integrin alphaVbeta3, file e2188be6-02b9-4564-e053-6605fe0a49d6
|
311
|
|
Determination of the binding epitope of RGD-peptidomimetics to αvβ3 and αIIbβ3 integrin-rich intact cells by NMR and computational studies, file e2188be6-041b-4564-e053-6605fe0a49d6
|
293
|
|
A Library Approach to the Development of BenzaPhos, Highly Efficient Chiral Supramolecular Ligands for Asymmetric Hydrogenation, file e2188be6-0267-4564-e053-6605fe0a49d6
|
247
|
|
SupraBox: a New Class of Chiral Supramolecular Oxazoline Ligands, file e2188be6-0268-4564-e053-6605fe0a49d6
|
196
|
|
Solid-phase synthesis of peptides containing reverse-turn mimetic bicyclic lactams, file e2188be5-fb89-4564-e053-6605fe0a49d6
|
99
|
|
Rh-Catalyzed Asymmetric Reactions with a Dynamic Library of Chiral Tropos Phosphorus Ligands, file e2188be6-76de-4564-e053-6605fe0a49d6
|
88
|
|
Kiss and Run: Promoting Effective and Targeted Cellular Uptake of a Drug Delivery Vehicle Composed of an Integrin-Targeting Diketopiperazine Peptidomimetic and a Cell-Penetrating Peptide, file e2188be7-3031-4564-e053-6605fe0a49d6
|
77
|
|
Synthesis and Conformational Studies of Peptidomimetics Containing a New Bifunctional Diketopiperazine Scaffold Acting as a β-Hairpin Inducer, file e2188be6-71c5-4564-e053-6605fe0a49d6
|
73
|
|
Discovery of a new efficient chiral ligand for copper-catalyzed enantioselective Michael additions by high-throughput screening of a parallel library, file e2188be5-fceb-4564-e053-6605fe0a49d6
|
69
|
|
Hydrogen-Bonding Donor/Acceptor Scales in b -Sulfonamidopeptides., file e2188be5-f7e5-4564-e053-6605fe0a49d6
|
67
|
|
Combinatorial libraries of chiral ligands for enantioselective catalysis, file e2188be5-fd0a-4564-e053-6605fe0a49d6
|
57
|
|
A New Method for the Solution and Solid Phase Synthesis of Chiral b-Sulfonopeptides Under Mild Conditions., file e2188be5-f7df-4564-e053-6605fe0a49d6
|
55
|
|
Synthesis of (S)- and (R)-5-oxo-piperazine-2-carboxylic acid and its application to peptidomimetics., file e2188be6-75db-4564-e053-6605fe0a49d6
|
49
|
|
Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin (V3), file e2188be7-61e5-4564-e053-6605fe0a49d6
|
47
|
|
Cyclative cleavage via solid-phase supported stabilized sulfur ylides: synthesis of macrocyclic lactones, file e2188be6-e81c-4564-e053-6605fe0a49d6
|
44
|
|
Synthetic studies on the sarcodictyins: synthesis of fully functionalized cyclization precursors, file e2188be5-fcf1-4564-e053-6605fe0a49d6
|
40
|
|
Synthesis and screening of new chiral ligands for the copper-catalysed enantioselective allylic substitution, file e2188be5-fcf6-4564-e053-6605fe0a49d6
|
37
|
|
Optimization of new chiral ligands for the copper-catalysed enantioselective conjugate addition of Et2Zn to nitroolefins by high-throughput screening of a parallel library, file e2188be5-fcf0-4564-e053-6605fe0a49d6
|
36
|
|
Synthesis of Combinatorial Libraries of Vinylogous Sulfonamidopeptides (Vs-Peptides)., file e2188be5-f7e3-4564-e053-6605fe0a49d6
|
32
|
|
Investigation of a New Family of Chiral Ligands for Enantioselective Catalysis via Parallel Synthesis and High-Throughput Screening., file e2188be5-f7e7-4564-e053-6605fe0a49d6
|
28
|
|
A Catalytic and Enantioselective Desymmetrization of Meso Cyclic Allylic Bisdiethylphosphates with Organozinc Reagents, file e2188be5-f9e6-4564-e053-6605fe0a49d6
|
28
|
|
A carbonylative cross-coupling strategy to the total synthesis of the sarcodictyins: preliminary studies and synthesis of a cyclization precursor, file e2188be5-fcef-4564-e053-6605fe0a49d6
|
28
|
|
Synthesis of (S)- and (R)-5-oxo-piperazine-2-carboxylic acid and its application to peptidomimetics., file e2188be5-fd5c-4564-e053-6605fe0a49d6
|
27
|
|
Redox Chemistry Associated with the Complexation of Vanadium (V) and Tungsten (VI) by meso-Octaethylporphyrinogen: Formation and Cleavage of Cyclopropane Units Functioning as Shuttles of two Electrons., file e2188be5-f7de-4564-e053-6605fe0a49d6
|
24
|
|
Enantioselective binding of dipeptides using acyclic receptors, file e2188be5-fce8-4564-e053-6605fe0a49d6
|
24
|
|
The Four-electron Oxidation of meso-Octaethylporphirinogen via a Metal-mediated Dealkylation Process: Formation of [RuL(PhCN)2] [H2L = 5,15-dihydro-5,5,10,15,20-hexaethylporphyrin]., file e2188be6-0070-4564-e053-6605fe0a49d6
|
21
|
|
Carbohydrate Metal Complexes as Ligands for Alkali Cations, file e2188be6-0071-4564-e053-6605fe0a49d6
|
21
|
|
A Trifunctional Steroid-Based Scaffold for Combinatorial Chemistry, file e2188be5-f9e4-4564-e053-6605fe0a49d6
|
20
|
|
Effect of ligands and additives on the palladium-promoted carbonylative coupling of vinyl stannanes and electron-poor enol triflates, file e2188be5-fce6-4564-e053-6605fe0a49d6
|
20
|
|
Combinatorial Libraries - Studies in Molecular Recognition and the Quest for New Catalysts., file e2188be5-f7e0-4564-e053-6605fe0a49d6
|
17
|
|
Synthetic Studies on Sarcodictyins and Eleutherobin: Synthesis of Fully Functionalized Cyclization Precursors, file e2188be5-fa3b-4564-e053-6605fe0a49d6
|
17
|
|
Synthesis, conformational studies and binding properties of acyclic receptors for N-protected amino acids and dipeptides, file e2188be5-fced-4564-e053-6605fe0a49d6
|
13
|
|
Foldamers of bifunctional diketopiperazines displaying a -bend ribbon structure., file e2188be5-fd5d-4564-e053-6605fe0a49d6
|
12
|
|
A combined fragment-based virtual screening and STD-NMR approach for the identification of E-cadherin ligands, file 00a105a3-acad-4267-be00-378b94953a61
|
11
|
|
Metallohosts Derived from the Assembly of Sugars Around Transition Metals - The Complexation of Alkali Metal Cations., file e2188be5-f7e1-4564-e053-6605fe0a49d6
|
11
|
|
Conformational switch and multiple supramolecular structures of a newly identified self-assembling protein-mimetic peptide from Pseudomonas aeruginosa YeaZ protein, file 0fdea102-aa5b-4098-a46d-81725f2d02a2
|
10
|
|
Discovery of a New Efficient Chiral Ligand for Copper Catalyzed Enantioselective Michael Additions by High-Throughput Screening of a Parallel Library, file e2188be5-f9e5-4564-e053-6605fe0a49d6
|
8
|
|
Copper phosphoramidite-catalyzed enantioselective desymmetrization of meso-cyclic allylic bisdiethyl phosphates, file e2188be5-fd0b-4564-e053-6605fe0a49d6
|
8
|
|
Transition Metal-Carbohydrate Chemistry. Part 2. Homoleptic Diacetoneglucose Complexes of Aluminium and Group 4 Metals., file e2188be6-006e-4564-e053-6605fe0a49d6
|
8
|
|
Insights into the Binding of Cyclic RGD Peptidomimetics to α5β1 Integrin by using Live-Cell NMR And Computational Studies, file e2188be6-cd67-4564-e053-6605fe0a49d6
|
7
|
|
Diacetoneglucose Complexes of Manganese(II) and Iron(II) and Their Organometallic Derivatization., file e2188be5-f7e4-4564-e053-6605fe0a49d6
|
6
|
|
Ureas: New Efficient Lewis Base Catalysts for the Allylation of Aldehydes, file e2188be5-fb82-4564-e053-6605fe0a49d6
|
6
|
|
Chiral (salen)Co(III)(N-benzyl-L-serine) derived phosphites: monodentate P-ligands for enantioselective catalytic applications, file e2188be5-fd58-4564-e053-6605fe0a49d6
|
6
|
|
PhthalaPhos: Chiral Supramolecular Ligands for Enantioselective Rhodium-Catalyzed Hydrogenation Reactions, file e2188be5-fd5e-4564-e053-6605fe0a49d6
|
6
|
|
Synthesis and Biological Evaluation of an isoDGR-Paclitaxel Conjugate Containing a Cell-Penetrating Peptide to Promote Cellular Uptake, file e2188be7-d0be-4564-e053-6605fe0a49d6
|
5
|
|
Optimizing the enzymatic release of MMAE from isoDGR-based small molecule drug conjugate by incorporation of a GPLG-PABC enzymatically cleavable linker, file 44716b1d-82af-45bd-a54f-45ec2965e74f
|
4
|
|
Transition Metal-Carbohydrate Chemistry. Part 4. Homoleptic Diacetoneglucose Complexes of Molybdenum and Tungsten: Chiral Ligands Associated to a M-M Triple Bond., file e2188be6-0072-4564-e053-6605fe0a49d6
|
4
|
|
Design, Synthesis and Catalytic Activity of (Cyclopentadienone)iron Complexes Containing a Stereogenic Plane and a Stereogenic Axis, file aa777344-6632-43c4-ade0-60c2a64295b7
|
3
|
|
Combination of a binaphthol-derived phosphite and a C1-symmetric phosphinamine generates heteroleptic catalysts in Rh- and Pd-mediated reactions, file e2188be5-fd5a-4564-e053-6605fe0a49d6
|
3
|
|
Acceleration of hemiacetal cleavage through hydrogen bonding : a new synthetic catalyst with balanced conformational flexibility and preorganization, file e2188be6-0052-4564-e053-6605fe0a49d6
|
3
|
|
Oxo and Imido Molybdenum (VI) and Tungsten (VI) Functionalities Supported by Diacetoneglucose, file e2188be6-0078-4564-e053-6605fe0a49d6
|
3
|
|
Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting, file e2188be6-f6fb-4564-e053-6605fe0a49d6
|
3
|
|
Investigating the interaction of cyclic RGD peptidomimetics with αVβ6integrin by biochemical and molecular docking studies, file e2188be6-fb26-4564-e053-6605fe0a49d6
|
3
|
|
Rational design of antiangiogenic helical oligopeptides targeting the vascular endothelial growth factor receptors, file e2188be7-406c-4564-e053-6605fe0a49d6
|
3
|
|
Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery, file e2188be7-49e9-4564-e053-6605fe0a49d6
|
3
|
|
Cyclic RGD and isoDGR Integrin Ligands Containing cis-2-amino-1-cyclopentanecarboxylic (cis-β-ACPC) Scaffolds, file e2188be7-9070-4564-e053-6605fe0a49d6
|
3
|
|
Optimizing the enzymatic release of MMAE from isoDGR-based small molecule drug conjugate by incorporation of a GPLG-PABC enzymatically cleavable linker, file f66959ec-33ec-4368-92df-5c3f1d7fafb8
|
3
|
|
Bifunctional 2,5-Diketopiperazines as Rigid Three-Dimensional Scaffolds in Receptors and Peptidomimetics, file e2188be5-fe26-4564-e053-6605fe0a49d6
|
2
|
|
Bifunctional 2,5-Diketopiperazines as Efficient Organocatalysts for the Enantioselective Conjugate Addition of Aldehydes to Nitroolefins, file e2188be5-fe29-4564-e053-6605fe0a49d6
|
2
|
|
Tumor Targeting with an isoDGR-Drug Conjugate, file e2188be6-fb20-4564-e053-6605fe0a49d6
|
2
|
|
Chiral Iron Complexes in Asymmetric Organic Transformations, file 20a3bea9-5e49-4086-99d9-1a925eb7471c
|
1
|
|
Multidisciplinary approaches in research and development of innovative drugs: project for an international collaborative training network.Ente finanaziatore: Fondazione CARIPLO, Bando "RST - Promuovere la formazione di capitale umano di eccellenza. Progetto in Partnership 2010"., file e2188be5-f844-4564-e053-6605fe0a49d6
|
1
|
|
Cyclic RGD-Peptidomimetics Containing Bifunctional Diketopiperazine Scaffolds as New Potent Integrin Ligands, file e2188be5-fd5b-4564-e053-6605fe0a49d6
|
1
|
|
Synthesis, Characterization, and Biological Evaluation of a Dual-Action Ligand Targeting αvβ3 Integrin and VEGF Receptors, file e2188be6-226b-4564-e053-6605fe0a49d6
|
1
|
|
Synthesis and biological evaluation of RGD peptidomimetic-paclitaxel conjugates bearing lysosomally cleavable linkers, file e2188be6-27b0-4564-e053-6605fe0a49d6
|
1
|
|
Efficient Synthesis of Amines by Iron-Catalyzed C=N Transfer Hydrogenation and C=O Reductive Amination, file e2188be7-1c6c-4564-e053-6605fe0a49d6
|
1
|
| Totale |
4.083 |