Sfoglia per Autore
Chiral (Cyclopentadienone)iron Complexes for the Catalytic Asymmetric Hydrogenation of Ketones
2015-01-01 Gajewski, Piotr; Renom Carrasco, Marc; Vailati Facchini, Sofia; Pignataro, Luca; Lefort, Laurent; de Vries, Johannes G.; Ferraccioli, Raffaella; Forni, Alessandra; Piarulli, Umberto; Gennari, Cesare
Cyclic isoDGR and RGD Peptidomimetics Containing Bifunctional Diketopiperazine Scaffolds are Integrin Antagonists
2015-01-01 Panzeri, Silvia; Zanella, Simone; Arosio, Daniela; Vahdati, Leila; Dal Corso, Alberto; Pignataro, Luca; Paolillo, Mayra; Schinelli, Sergio; Belvisi, Laura; Gennari, Cesare; Piarulli, Umberto
Synthesis, Characterization, and Biological Evaluation of a Dual-Action Ligand Targeting αvβ3 Integrin and VEGF Receptors
2015-01-01 Zanella, Simone; Mingozzi, Michele; Dal Corso, Alberto; Fanelli, Roberto; Arosio, Daniela; Cosentino, Marco; Schembri, Laura; Marino, Franca; De Zotti, Marta; Formaggio, Fernando; Pignataro, Luca; Belvisi, Laura; Piarulli, Umberto; Gennari, Cesare
Assisted Tandem Catalysis: Metathesis Followed by Asymmetric Hydrogenation from a Single Ruthenium Source
2015-01-01 Renom-Carrasco, M.; Gajewski, P.; Pignataro, L.; Devries, J. G.; Piarulli, U.; Gennari, C.; Lefort, L.
Synthesis and biological evaluation of RGD peptidomimetic-paclitaxel conjugates bearing lysosomally cleavable linkers
2015-01-01 Dal Corso, Alberto; Caruso, Michele; Belvisi, Laura; Arosio, Daniela; Piarulli, Umberto; Albanese, Clara; Gasparri, Fabio; Marsiglio, Aurelio; Sola, Francesco; Troiani, Sonia; Valsasina, Barbara; Pignataro, Luca; Donati, Daniele; Gennari, Cesare
Synthesis of (R)-BINOL-Derived (Cyclopentadienone)iron Complexes and Their Application in the Catalytic Asymmetric Hydrogenation of Ketones
2015-01-01 Gajewski, P.; Renom-Carrasco, M.; Facchini, S. V.; Pignataro, L.; Lefort, L.; De Vries, J. G.; Ferraccioli, R.; Piarulli, U.; Gennari, C.
Computational design of novel peptidomimetic inhibitors of cadherin homophilic interactions
2015-01-01 Doro, Fabio; Colombo, Cinzia; Alberti, Chiara; Arosio, Daniela; Belvisi, Laura; Casagrande, Cesare; Fanelli, Roberto; Manzoni, Leonardo; Parisini, Emilio; Piarulli, Umberto; Luison, Elena; Figini, Mariangela; Tomassetti, Antonella; Civera, Monica
Synthesis and conformational studies of a stable peptidomimetic β-hairpin based on a bifunctional diketopiperazine turn inducer
2015-01-01 Vahdati, Leila; Fanelli, Roberto; Bernadat, Guillaume; Correia, Isabelle; Lequin, Olivier; Ongeri, Sandrine; Piarulli, Umberto
Asymmetric Transfer Hydrogenation of Ketones with Modified Grubbs Metathesis Catalysts: On the Way to a Tandem Process
2016-01-01 Renom Carrasco, Marc; Gajewski, Piotr; Pignataro, Luca; De Vries, Johannes G.; Piarulli, Umberto; Gennari, Cesare; Lefort, Laurent
A Mixed Ligand Approach for the Asymmetric Hydrogenation of 2-Substituted Pyridinium Salts
2016-01-01 Renom Carrasco, Marc; Gajewski, Piotr; Pignataro, Luca; de Vries, Johannes G.; Piarulli, Umberto; Gennari, Cesare; Lefort, Laurent
Expanding the Catalytic Scope of (Cyclopentadienone)iron Complexes to the Hydrogenation of Activated Esters to Alcohols
2016-01-01 Gajewski, Piotr; Gonzalez de Castro, Angela; Renom Carrasco, Marc; Piarulli, Umberto; Gennari, Cesare; de Vries, Johannes G.; Lefort, Laurent; Pignataro, Luca
Asymmetric Hydrogenation of 3-Substituted Pyridinium Salts
2016-01-01 Renom Carrasco, Marc; Gajewski, Piotr; Pignataro, Luca; de Vries, Johannes G.; Piarulli, Umberto; Gennari, Cesare; Lefort, Laurent
Enantioselective reductions promoted by (cyclopentadienone)iron complexes
2017-01-01 Piarulli, Umberto; Fachini, Sofia Vailati; Pignataro, Luca
Tumor Targeting with an isoDGR-Drug Conjugate
2017-01-01 Zanella, S.; Angerani, S.; Pina, A.; López Rivas, P.; Giannini, C.; Panzeri, S.; Arosio, D.; Caruso, M.; Gasparri, F.; Fraietta, I.; Albanese, C.; Marsiglio, A.; Pignataro, L.; Belvisi, L.; Piarulli, Umberto; Gennari, C.
Insights into the Binding of Cyclic RGD Peptidomimetics to α5β1 Integrin by using Live-Cell NMR And Computational Studies
2017-01-01 Guzzetti, Ileana; Civera, Monica; Vasile, Francesca; Arosio, Daniela; Tringali, Cristina; Piarulli, Umberto; Gennari, Cesare; Pignataro, Luca; Belvisi, Laura; Potenza, Donatella
Investigating the interaction of cyclic RGD peptidomimetics with αVβ6integrin by biochemical and molecular docking studies
2017-01-01 Civera, Monica; Arosio, Daniela; Bonato, Francesca; Manzoni, Leonardo; Pignataro, Luca; Zanella, Simone; Gennari, Cesare; Piarulli, Umberto; Belvisi, Laura
Synthesis and Characterization of Hairpin Mimics that Modulate the Early Oligomerization and Fibrillization of Amyloid β-Peptide
2017-01-01 Vahdati, Leila; Kaffy, Julia; Brinet, Dimitri; Bernadat, Guillaume; Correia, Isabelle; Panzeri, Silvia; Fanelli, Roberto; Lequin, Olivier; Taverna, Myriam; Ongeri, Sandrine; Piarulli, Umberto
Synthesis of [Bis(hexamethylene)cyclopentadienone]iron Tricarbonyl and its Application to the Catalytic Reduction of C=O Bonds
2017-01-01 VAILATI FACCHINI, Sofia; Neudörfl, Jörg Martin; Pignataro, Luca; Cettolin, Mattia; Gennari, Cesare; Berkessel, Albrecht; Piarulli, Umberto
Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting
2018-01-01 BODERO PADILLA, LIZETH ALICIA; Rivas, Paula López; Korsak, Barbara; Hechler, Torsten; Pahl, Andreas; Müller, Christoph; Arosio, Daniela; Pignataro, LUCA LUIGI; Gennari, CESARE MARIO ARTURO; Piarulli, Umberto
Efficient Synthesis of Amines by Iron-Catalyzed C=N Transfer Hydrogenation and C=O Reductive Amination
2018-01-01 Facchini, Sofia Vailati; Cettolin, Mattia; Bai, Xishan; Casamassima, Giuseppe; Pignataro, Luca; Gennari, Cesare; Piarulli, Umberto
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
Chiral (Cyclopentadienone)iron Complexes for the Catalytic Asymmetric Hydrogenation of Ketones | 1-gen-2015 | Gajewski, Piotr; Renom Carrasco, Marc; Vailati Facchini, Sofia; Pignataro, Luca; Lefort, Laurent; de Vries, Johannes G.; Ferraccioli, Raffaella; Forni, Alessandra; Piarulli, Umberto; Gennari, Cesare | |
Cyclic isoDGR and RGD Peptidomimetics Containing Bifunctional Diketopiperazine Scaffolds are Integrin Antagonists | 1-gen-2015 | Panzeri, Silvia; Zanella, Simone; Arosio, Daniela; Vahdati, Leila; Dal Corso, Alberto; Pignataro, Luca; Paolillo, Mayra; Schinelli, Sergio; Belvisi, Laura; Gennari, Cesare; Piarulli, Umberto | |
Synthesis, Characterization, and Biological Evaluation of a Dual-Action Ligand Targeting αvβ3 Integrin and VEGF Receptors | 1-gen-2015 | Zanella, Simone; Mingozzi, Michele; Dal Corso, Alberto; Fanelli, Roberto; Arosio, Daniela; Cosentino, Marco; Schembri, Laura; Marino, Franca; De Zotti, Marta; Formaggio, Fernando; Pignataro, Luca; Belvisi, Laura; Piarulli, Umberto; Gennari, Cesare | |
Assisted Tandem Catalysis: Metathesis Followed by Asymmetric Hydrogenation from a Single Ruthenium Source | 1-gen-2015 | Renom-Carrasco, M.; Gajewski, P.; Pignataro, L.; Devries, J. G.; Piarulli, U.; Gennari, C.; Lefort, L. | |
Synthesis and biological evaluation of RGD peptidomimetic-paclitaxel conjugates bearing lysosomally cleavable linkers | 1-gen-2015 | Dal Corso, Alberto; Caruso, Michele; Belvisi, Laura; Arosio, Daniela; Piarulli, Umberto; Albanese, Clara; Gasparri, Fabio; Marsiglio, Aurelio; Sola, Francesco; Troiani, Sonia; Valsasina, Barbara; Pignataro, Luca; Donati, Daniele; Gennari, Cesare | |
Synthesis of (R)-BINOL-Derived (Cyclopentadienone)iron Complexes and Their Application in the Catalytic Asymmetric Hydrogenation of Ketones | 1-gen-2015 | Gajewski, P.; Renom-Carrasco, M.; Facchini, S. V.; Pignataro, L.; Lefort, L.; De Vries, J. G.; Ferraccioli, R.; Piarulli, U.; Gennari, C. | |
Computational design of novel peptidomimetic inhibitors of cadherin homophilic interactions | 1-gen-2015 | Doro, Fabio; Colombo, Cinzia; Alberti, Chiara; Arosio, Daniela; Belvisi, Laura; Casagrande, Cesare; Fanelli, Roberto; Manzoni, Leonardo; Parisini, Emilio; Piarulli, Umberto; Luison, Elena; Figini, Mariangela; Tomassetti, Antonella; Civera, Monica | |
Synthesis and conformational studies of a stable peptidomimetic β-hairpin based on a bifunctional diketopiperazine turn inducer | 1-gen-2015 | Vahdati, Leila; Fanelli, Roberto; Bernadat, Guillaume; Correia, Isabelle; Lequin, Olivier; Ongeri, Sandrine; Piarulli, Umberto | |
Asymmetric Transfer Hydrogenation of Ketones with Modified Grubbs Metathesis Catalysts: On the Way to a Tandem Process | 1-gen-2016 | Renom Carrasco, Marc; Gajewski, Piotr; Pignataro, Luca; De Vries, Johannes G.; Piarulli, Umberto; Gennari, Cesare; Lefort, Laurent | |
A Mixed Ligand Approach for the Asymmetric Hydrogenation of 2-Substituted Pyridinium Salts | 1-gen-2016 | Renom Carrasco, Marc; Gajewski, Piotr; Pignataro, Luca; de Vries, Johannes G.; Piarulli, Umberto; Gennari, Cesare; Lefort, Laurent | |
Expanding the Catalytic Scope of (Cyclopentadienone)iron Complexes to the Hydrogenation of Activated Esters to Alcohols | 1-gen-2016 | Gajewski, Piotr; Gonzalez de Castro, Angela; Renom Carrasco, Marc; Piarulli, Umberto; Gennari, Cesare; de Vries, Johannes G.; Lefort, Laurent; Pignataro, Luca | |
Asymmetric Hydrogenation of 3-Substituted Pyridinium Salts | 1-gen-2016 | Renom Carrasco, Marc; Gajewski, Piotr; Pignataro, Luca; de Vries, Johannes G.; Piarulli, Umberto; Gennari, Cesare; Lefort, Laurent | |
Enantioselective reductions promoted by (cyclopentadienone)iron complexes | 1-gen-2017 | Piarulli, Umberto; Fachini, Sofia Vailati; Pignataro, Luca | |
Tumor Targeting with an isoDGR-Drug Conjugate | 1-gen-2017 | Zanella, S.; Angerani, S.; Pina, A.; López Rivas, P.; Giannini, C.; Panzeri, S.; Arosio, D.; Caruso, M.; Gasparri, F.; Fraietta, I.; Albanese, C.; Marsiglio, A.; Pignataro, L.; Belvisi, L.; Piarulli, Umberto; Gennari, C. | |
Insights into the Binding of Cyclic RGD Peptidomimetics to α5β1 Integrin by using Live-Cell NMR And Computational Studies | 1-gen-2017 | Guzzetti, Ileana; Civera, Monica; Vasile, Francesca; Arosio, Daniela; Tringali, Cristina; Piarulli, Umberto; Gennari, Cesare; Pignataro, Luca; Belvisi, Laura; Potenza, Donatella | |
Investigating the interaction of cyclic RGD peptidomimetics with αVβ6integrin by biochemical and molecular docking studies | 1-gen-2017 | Civera, Monica; Arosio, Daniela; Bonato, Francesca; Manzoni, Leonardo; Pignataro, Luca; Zanella, Simone; Gennari, Cesare; Piarulli, Umberto; Belvisi, Laura | |
Synthesis and Characterization of Hairpin Mimics that Modulate the Early Oligomerization and Fibrillization of Amyloid β-Peptide | 1-gen-2017 | Vahdati, Leila; Kaffy, Julia; Brinet, Dimitri; Bernadat, Guillaume; Correia, Isabelle; Panzeri, Silvia; Fanelli, Roberto; Lequin, Olivier; Taverna, Myriam; Ongeri, Sandrine; Piarulli, Umberto | |
Synthesis of [Bis(hexamethylene)cyclopentadienone]iron Tricarbonyl and its Application to the Catalytic Reduction of C=O Bonds | 1-gen-2017 | VAILATI FACCHINI, Sofia; Neudörfl, Jörg Martin; Pignataro, Luca; Cettolin, Mattia; Gennari, Cesare; Berkessel, Albrecht; Piarulli, Umberto | |
Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting | 1-gen-2018 | BODERO PADILLA, LIZETH ALICIA; Rivas, Paula López; Korsak, Barbara; Hechler, Torsten; Pahl, Andreas; Müller, Christoph; Arosio, Daniela; Pignataro, LUCA LUIGI; Gennari, CESARE MARIO ARTURO; Piarulli, Umberto | |
Efficient Synthesis of Amines by Iron-Catalyzed C=N Transfer Hydrogenation and C=O Reductive Amination | 1-gen-2018 | Facchini, Sofia Vailati; Cettolin, Mattia; Bai, Xishan; Casamassima, Giuseppe; Pignataro, Luca; Gennari, Cesare; Piarulli, Umberto |
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