BROGGINI, GIANLUIGI
 Distribuzione geografica
Continente #
NA - Nord America 13.002
EU - Europa 5.742
AS - Asia 3.156
SA - Sud America 392
AF - Africa 34
Continente sconosciuto - Info sul continente non disponibili 16
OC - Oceania 6
Totale 22.348
Nazione #
US - Stati Uniti d'America 12.869
IT - Italia 2.546
SG - Singapore 1.066
UA - Ucraina 1.020
CN - Cina 528
TR - Turchia 519
SE - Svezia 471
HK - Hong Kong 407
VN - Vietnam 407
BR - Brasile 338
DE - Germania 338
GB - Regno Unito 337
FI - Finlandia 294
IE - Irlanda 291
RU - Federazione Russa 166
IN - India 77
CA - Canada 67
FR - Francia 67
JP - Giappone 67
MX - Messico 54
ES - Italia 48
PL - Polonia 31
ZA - Sudafrica 25
BD - Bangladesh 22
NL - Olanda 22
AR - Argentina 18
BE - Belgio 18
CH - Svizzera 17
EU - Europa 16
IQ - Iraq 16
CZ - Repubblica Ceca 15
AT - Austria 13
VE - Venezuela 10
AE - Emirati Arabi Uniti 8
LT - Lituania 8
PT - Portogallo 8
EC - Ecuador 7
RO - Romania 7
AU - Australia 6
ID - Indonesia 6
NO - Norvegia 6
IL - Israele 5
BG - Bulgaria 4
PE - Perù 4
PY - Paraguay 4
BB - Barbados 3
CL - Cile 3
CO - Colombia 3
DK - Danimarca 3
GR - Grecia 3
JO - Giordania 3
PK - Pakistan 3
SA - Arabia Saudita 3
UY - Uruguay 3
AZ - Azerbaigian 2
BO - Bolivia 2
DM - Dominica 2
DZ - Algeria 2
HN - Honduras 2
MY - Malesia 2
PA - Panama 2
TN - Tunisia 2
AL - Albania 1
BH - Bahrain 1
BN - Brunei Darussalam 1
BT - Bhutan 1
BY - Bielorussia 1
EG - Egitto 1
ET - Etiopia 1
GA - Gabon 1
GD - Grenada 1
GT - Guatemala 1
HU - Ungheria 1
IR - Iran 1
KG - Kirghizistan 1
KZ - Kazakistan 1
LB - Libano 1
LU - Lussemburgo 1
MA - Marocco 1
MD - Moldavia 1
ME - Montenegro 1
MM - Myanmar 1
MO - Macao, regione amministrativa speciale della Cina 1
NP - Nepal 1
OM - Oman 1
RS - Serbia 1
SI - Slovenia 1
SK - Slovacchia (Repubblica Slovacca) 1
SN - Senegal 1
TH - Thailandia 1
TJ - Tagikistan 1
TT - Trinidad e Tobago 1
TW - Taiwan 1
UZ - Uzbekistan 1
Totale 22.348
Città #
Dallas 1.898
Milan 1.738
Fairfield 1.649
Ashburn 962
Woodbridge 927
Jacksonville 780
Houston 682
Seattle 669
Chandler 628
Singapore 623
Wilmington 562
Cambridge 506
Hong Kong 407
Ann Arbor 391
Dearborn 378
Dublin 291
Princeton 280
Nyköping 279
Izmir 224
Dong Ket 211
Boardman 187
Beijing 171
Rome 132
The Dalles 125
Los Angeles 121
San Mateo 109
Chicago 103
San Diego 97
New York 81
Como 74
London 72
Santa Clara 66
Munich 63
Tokyo 63
Ogden 55
Kocaeli 50
São Paulo 49
Kunming 33
Mexico City 33
Düsseldorf 32
Ho Chi Minh City 32
Turku 32
Washington 32
Hefei 31
Buffalo 30
Des Moines 30
Montreal 29
Verona 28
Warsaw 26
Atlanta 25
Chennai 25
Phoenix 25
Orem 24
Boston 22
Johannesburg 22
Stockholm 21
Brooklyn 19
Denver 19
Manchester 19
Nanjing 18
Toronto 18
Mumbai 17
Nanchang 17
Council Bluffs 16
Hanoi 16
Norwalk 16
Brussels 15
Helsinki 14
Brno 13
Clausthal-Zellerfeld 13
Paris 13
Berlin 12
Frankfurt am Main 12
Fuzhou 12
Jinan 12
Poplar 12
Rio de Janeiro 12
San Francisco 12
West Jordan 12
Amsterdam 11
Guangzhou 11
Kilburn 11
Vienna 11
Elk Grove Village 10
Bari 9
Campinas 9
Chiswick 9
Hounslow 9
New Delhi 9
Nuremberg 9
Philadelphia 9
Rotonda 9
Ankara 8
Auburn Hills 8
Belo Horizonte 8
Dhaka 8
Edinburgh 8
New Bedfont 8
Pisa 8
Salt Lake City 8
Totale 16.764
Nome #
1,3-Dipolar cycloadditions to nitrogen-substituted allenes 1.174
1,3-Dipolar cycloadditions to allenes 1.122
Boehmeriasin A as new lead compound for the inhibition of topoisomerases and SIRT2 236
C-C, C-O, C-N Bond Formation on sp2-Carbon by Pd(II)-Catalyzed Reactions Involving Oxidant Agents 226
A facile synthesis of flumazenil analogues 209
Copper(II)-catalyzed alkoxyhalogenation of alkynyl ureas and amides as a route to haloalkylidene substituted heterocycles 208
(Diacyloxyiodo)benzenes-Driven Palladium-Catalyzed Cyclizations of Unsaturated N-Sulfonylamides: Opportunities of Path Selection 199
A synthetic route to [1,2,4]triazolo[1,5-a][4,1]benzoxazepines 196
A New Entry to [1,2,4]Triazolo[1,5-a][1,4]benzodiazepin-6-ones via Intramolecular Nitrilimine Cycloaddition to the Cyano Group 195
An alternative synthesis of 2-alkylidene-3,4-dihydro-2H-1,4-benzoxazines by intramolecular gold-catalyzed hydroalkoxylation of 2-(prop-2-yn-1-ylamino)-phenols 192
Intramolecular Oxidative Palladium-Catalyzed Amination Involving Double C-H Functionalization of Unactivated Olefins 192
Palladium-catalyzed domino carbopalladation/5-exo-allylic amination of α-amino allenamides: an efficient entry to enantiopure imidazolidinones 190
Synthesis and biological evaluation of 1,7,8,8a-tetrahydro-3H-oxazolo[3,4-a]pyrazin-6(5H)-ones as antitumoral agents 190
Stereoselective intramolecular cycloadditions of homochiral nitrile imines: synthesis of enantiomerically pure 3,3a-dihydro-pyrazolo[1,5-a][1,4] benzodiazepine-6(4H)-ones 190
Synthesis of Pironetin-Dumetorine Hybrids as Tubulin Binders 189
Access to pyrrolo-pyridines by gold-catalyzed hydroarylation of pyrroles tethered to terminal alkynes 186
SYNTHESIS OF ENANTIOPURE 4-AMINO-3-HYDROXYMETHYL-TETRAHYDROQUINOLINES VIA AN INTRAMOLECULAR NITRONE CYCLOADDITION 180
Selective intramolecular palladium(II)-catalyzed aminooxygenation vs. diamination of alkenylureas: efficient microwave-assisted reactions to bicyclic piperazinones 178
Ruthenium-Catalyzed Hydroamination of Aminoallenes: an Approach to Vinyl Substituted Heterocycles 178
A valuable approach to enantiopure partially saturated pyrrolo- and indolo[1,2-a]indoles by intramolecular nitrone cycloadditions to the cyclohexene ring 177
Dipolarophilic behavior of the isoxazole ring in intramolecular nitrilimine cycloadditions 175
5-Heterosubstituted 4-methylene-4,5-dihydroisoxazoles: Ready accessibility and versatile reactivity 175
Intra-Intermolecular Palladium-Catalyzed Domino Reactions of Glycine Allylamides for the Synthesis of Diversely Functionalized Piperazinones 172
Synthesis of 1,4-benzodiazepinones via palladium-catalysed allene carbopalladation/amination domino sequence 171
Palladium-Catalysed Carbo- and Hydroamination of Allenyl Ethers and Aminoallenes: Available Entry to Nitrogen-Containing Benzo-Fused Rings 171
Palladium(II)/copper halide/solvent combination for selective intramolecular domino reactions of indole carboxylic acid allylamides. An unprecedented arylation/esterification sequence 168
Solvent- and ligand-free palladium-catalyzed amination of aryl halides 168
Dehydrogenative Allylic Aminations of But-3-enoic Acid Derivatives 166
Efficient Approach to the Unknown Isoxazolo[3,4-d]thieno[2,3-b]pyridine System by Regioselective Intramolecular Nitrone Cycloadditions 165
The intramolecular azide cycloaddition route to triazolam analogues 165
New Mechanistic Evidence on the Reaction between Sulfonylallenes and Nitrile Oxides 164
Synthesis of enantiopure 3-hydroxymethylchromanes via intramolecular nitrone cycloaddition 162
N,N-Disubstituted Propargylamines as Tools in the Sequential 1,3-Dipolar Cycloaddition/Arylation Processes to the Formation of Polyheterocyclic Systems 162
Transition metal complexation in 1,3-dipolar cycloadditions 162
Diastereoselective synthesis of bis(3,5)pyrazolophanes by sequential inter- and intramolecular cycloadditions of homochiral nitrilimines 161
Recent advances in heterobimetallic palladium(ii)/copper(ii) catalyzed domino difunctionalization of carbon–carbon multiple bonds 161
Intramolecular Aminoazidation of Unactivated Terminal Alkenes by Palladium-Catalyzed Reactions with Hydrogen Peroxide as the Oxidant 160
Intramolecular oxidative palladium-catalyzed diamination reactions of alkenyl sulfamates: an efficient synthesis of [1,2,5]thiadiazolo-fused piperazinones 159
Transition metal-catalyzed hydroamination and carboamination reactions of anthranilic allenamides as a route to 2-vinyl- and 2-(a-styryl)-quinazolin-4-one derivatives 158
New Access to Kainic Acid via Intramolecular Palladium-Catalyzed Allylic Alkylation 157
Intramolecular azide cycloadditions leading to [1,2,3]triazolo[1,5-a]quinoxalines 157
A valuable heterocyclic ring transformation: from isoxazolin-5(2H)-ones to quinolines 155
Palladium-Catalyzed Cyclization/Carbonylation as a Direct Route to 4-[(Methoxycarbonyl)methyl]-3,4-dihydroisoquinolinones 155
Synthesis of Bis-(3,5)pyrazolophanes by Sequential Intermolecular-Intramolecular Nitrilimine Cycloadditions 154
Intramolecular oxidative Pd(II)-catalyzed alkoxylation of 3-aza-5-alkenols with O2 as sole oxidant: mild conditions for the synthesis of 1,4-oxazine derivatives 154
Chimica degli eterocicli 153
Thermal behaviour of dipolarophile-containing acyl azides: intramolecular cycloaddition versus Curtius rearrangement 153
Uncommon intramolecular palladium-catalyzed cyclization of indole derivatives 152
A new synthesis of flumazenil suitable for fluorine-18 labeling 152
L-alanine benzylester as chiral inductor: Synthesis of enantiopure pyrazolo[1,5-a]-[1,4]benzodiazepine-4-ones via intramolecular nitrilimine cycloadditions 152
Pyrrolizidine and indolizidine syntheses involving 1,3-dipolar cycloadditions 152
Palladium-Catalyzed dual C-H or N-H functionalization of unfunctionalized indole derivatives with alkenes and arenes 152
A new protocol for the conversion of isoxazolidines to 1,3-aminoalcohols 151
Stereoselective intramolecular cycloadditions of homochiral N-alkenoyl aryl azides 150
Synthetic approach to imidazo[1,2-a]pyridine derivatives by the intramolecular nitrone cycloaddition methodology 150
Intramolecular Palladium-Catalyzed Aminocarboxylation of Olefins as a Direct Route to Bicyclic Oxazolidinones 150
Regiochemical aspects of intramolecular cycloadditions of nitrones derived from N-(2-alkenyl)-2-pyrrolecarbaldehydes. Competitive entries to pyrrolizidine and indolizidine derivatives 149
Intramolecular Cycloadditions of Nitrones Derived from 1-Allyl-2-pyrrolecarbaldehyde as a Route to Racemic and Enantiopure Pyrrolizidines and Indolizidines 148
Palladium-catalyzed C-N bond formation via direct C-H bond functionalization. Recent developments in heterocyclic synthesis 147
Enantiopure 2-piperidylacetaldehyde as useful building block in the diversity-oriented synthesis of polycyclic piperidine derivatives 147
The first case of asymmetric induction in intramolecular nitrile imine cycloadditions: synthesis of enantiopure 3-substituted 6-oxo-2,3,3a,5-tetrahydro-4-carbomethoxy-furo[3,4-c]pyrazoles 146
Dipolarophilic behaviour of (arylsulfonyl)allenes towards nitrilimines 146
Pd-Catalyzed Intramolecular Cyclization of Pyrrolo-2-carboxamides: Regiodivergent Routes to Pyrrolo-pyrazines and Pyrrolo-pyridines 146
Enantioselective intramolecular nitrone cycloaddition route to 3-(trifluoromethyl)-isoxazolidino[4,3-c]-chroman-4-ones and -quinolin-4-ones 146
Intramolecular Pd(II)-Catalyzed Cyclization of Propargylamides: Straightforward Synthesis of 5-Oxazole-carbaldehydes 145
Solvent-free, microwave-assisted N-arylation of indolines by using low palladium catalyst loadings 145
Regioselective Intramolecular Cycloaddition of C-(1-Acryloyl-2-pyrrolyl)-N-benzylnitrone: Entry to 6-Hydroxy-5-oxoindolizidines 144
Dipolarophilic behaviour of the thiophene ring in intramolecular nitrile imine cycloadditions 144
Regioselectivity on the palladium-catalyzed intramolecular cyclization of indole derivatives 142
A Valuable Synthesis of Pyrrolo[1,2-a]quinoxalines, Indolo[1,2-a]quinoxalines and their Aza-Analogues by Palladium-Catalyzed Intramolecular Carbon-Nitrogen Bond Formation 142
Selective 7- endo -Cyclization of 3-Aza-5-alkenols through Oxidative Pd(II)-Catalyzed Olefin Oxyarylation 142
Synthesis of tetrazolo[1,5-a][1,4]benzodiazepin-6-ones via intramolecular azide cycloadditions onto the cyano group 142
Palladium-mediated Approach to Dibenzo[b,e][1,4]diazepines and Benzopyrido-analogues. An Efficient Synthesis of Tarpane 141
Synthesis of enantiopure pyrrolo[3,4-c]pyrazole derivatives via intramolecular cycloaddition of homochiral nitrilimines 140
Synthesis of pyrazolo[1,5-a]quinoxalines 137
Relative and absolute stereocontrol in intramolecular nitrone cycloadditions to the cyclohexene ring 137
Access to pyrralo- and pyrido[1,2-a]indole derivatives by intramolecular nitrone cycloadditions. Effect of steric factors on the regioselective product formation 136
Nitrilimine cycloadditions onto partially saturated furo[3,4-c]thieno[2,3-d]pyrazoles. A problem in site selectivity 136
Intramolecular nitrile imide cycloadditions onto the furan ring: synthesis of the new 3a,4-dihydro-6H-difuro[3,2-c;3,4-d]pyrazole skeleton 136
Synthesis and Biological Evaluation of Migrastatin Macrotriazoles 136
A facile synthesis of 2-methyl-1,4-benzodiazepin-5-ones via intramolecular azide cycloaddition 135
Synthesis of enantiopure 4-amino-6-fluoro-3-(hydroxymethyl)chromanes via intramolecular nitrone cycloadditions 135
Oxidative cleavage of the isoxazolidine ring 134
Access to a Novel Class of Tetracyclic 1,4-Benzodiazepin-5-ones Starting from alpha-Aminoacids by Pd-Catalyzed Amination/1,3-Dipolar Cycloaddition as Key Steps 134
Intramolecular cycloadditions of N-alkenoyl aryl azides 132
Nitrilimine cycloadditions in aqueous media 132
Intramolecular Azide Cycloaddition en Route to the New Pyrrolo[2,1-c][1,2,3]triazolo[1,5-a][1,4]benzodiazepine Skeleton 132
Iodoamination of Alkenyl Sulfonamides by Potassium Iodide and Hydrogen Peroxide in Aqueous Medium 132
Novel aspects of the silver carbonate promoted reaction of hydrazonyl chlorides with homoallylic and homopropargylic alcohols 131
Synthesis of N-(5-amino-2-pyrimidyl)-N '-[4-(p-fluorophenyl)-4-oxobutyl]piperazine, a useful intermediate to antipsychotic agents 130
Asymmetric induction by the (S)-1-phenylethyl group in intramolecular nitrile imine cycloadditions giving enantiopure 3,3a-dihydro-pyrazolo[1,5-alpha][1,4]benzodiazepine-4(6H)-ones 130
Divergent Palladium- and Platinum-Catalyzed Intramolecular Hydroamination/Hydroarylation of O-Propargyl-2-aminophenols 130
Diastereoselective nitrilimine cycloaddition to the C = N bond of enantiopure 1,4-benzodiazepinones 129
Intramolecular cycloadditions of nitrones derived from optically active 1-alkenyl-2-imidazolecarbaldehydes: regio- and diastereoselectivity 129
Synthesis of 5-hydroxymethyl-1,4-dioxan-2-one 129
Tunable Pd-Catalyzed Cyclization of Indole-2-carboxylic Acid Allenamides: Carboamination vs Microwave-Assisted Hydroamination 129
Efficient Synthesis of N-Methoxyindoles via Alkylative Cycloaddition of Nitrosoarenes with Alkynes 128
Copper-Catalyzed Alkoxylation as Key Step to Convert Isatin to Oxazinoindol-2-one Derivatives 127
Pd-Catalyzed Cyclization of 1-Allyl-2-indolecarboxamides by Intramolecular Amidation of Unactivated Ethylenic Bond 126
Acid-mediated decarboxylative C-H coupling between arenes and O-allyl carbamates 126
Totale 17.581
Categoria #
all - tutte 88.266
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 88.266


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/20211.670 0 0 0 0 0 262 162 203 330 181 203 329
2021/20221.507 172 316 115 34 32 46 139 56 73 198 152 174
2022/20231.883 230 89 135 186 138 412 14 272 226 53 75 53
2023/20243.001 422 400 462 598 628 188 34 57 89 28 27 68
2024/20252.165 52 39 446 47 62 112 61 127 229 142 188 660
2025/20264.431 414 689 1.460 887 648 333 0 0 0 0 0 0
Totale 22.592