BROGGINI, GIANLUIGI
 Distribuzione geografica
Continente #
NA - Nord America 14.166
EU - Europa 5.960
AS - Asia 4.146
SA - Sud America 423
AF - Africa 73
Continente sconosciuto - Info sul continente non disponibili 16
OC - Oceania 6
Totale 24.790
Nazione #
US - Stati Uniti d'America 14.016
IT - Italia 2.580
SG - Singapore 1.343
UA - Ucraina 1.021
CN - Cina 878
VN - Vietnam 636
TR - Turchia 522
SE - Svezia 472
HK - Hong Kong 447
GB - Regno Unito 354
BR - Brasile 352
DE - Germania 351
FI - Finlandia 297
IE - Irlanda 292
FR - Francia 203
RU - Federazione Russa 169
IN - India 99
CA - Canada 70
JP - Giappone 70
MX - Messico 65
ES - Italia 48
PL - Polonia 33
BD - Bangladesh 32
ZA - Sudafrica 31
IQ - Iraq 27
NL - Olanda 25
AR - Argentina 22
BE - Belgio 19
CH - Svizzera 17
EU - Europa 16
CZ - Repubblica Ceca 15
NG - Nigeria 15
AT - Austria 13
VE - Venezuela 13
AE - Emirati Arabi Uniti 9
ID - Indonesia 9
PK - Pakistan 9
EC - Ecuador 8
LT - Lituania 8
PT - Portogallo 8
SA - Arabia Saudita 8
RO - Romania 7
TN - Tunisia 7
AU - Australia 6
NO - Norvegia 6
CL - Cile 5
CO - Colombia 5
IL - Israele 5
NP - Nepal 5
PE - Perù 5
PY - Paraguay 5
UZ - Uzbekistan 5
AZ - Azerbaigian 4
BG - Bulgaria 4
JO - Giordania 4
MY - Malesia 4
PH - Filippine 4
TH - Thailandia 4
TW - Taiwan 4
UY - Uruguay 4
BB - Barbados 3
BO - Bolivia 3
DK - Danimarca 3
EG - Egitto 3
GR - Grecia 3
KE - Kenya 3
KZ - Kazakistan 3
MA - Marocco 3
PA - Panama 3
ZW - Zimbabwe 3
AL - Albania 2
DM - Dominica 2
DZ - Algeria 2
GT - Guatemala 2
HN - Honduras 2
HU - Ungheria 2
LB - Libano 2
OM - Oman 2
PS - Palestinian Territory 2
SN - Senegal 2
BH - Bahrain 1
BN - Brunei Darussalam 1
BT - Bhutan 1
BY - Bielorussia 1
CI - Costa d'Avorio 1
ET - Etiopia 1
GA - Gabon 1
GD - Grenada 1
GY - Guiana 1
HR - Croazia 1
IR - Iran 1
KG - Kirghizistan 1
LU - Lussemburgo 1
MD - Moldavia 1
ME - Montenegro 1
ML - Mali 1
MM - Myanmar 1
MO - Macao, regione amministrativa speciale della Cina 1
QA - Qatar 1
RS - Serbia 1
Totale 24.785
Città #
Dallas 1.906
Milan 1.748
Fairfield 1.649
Ashburn 1.049
Woodbridge 927
San Jose 801
Singapore 796
Jacksonville 780
Houston 684
Seattle 669
Chandler 628
Wilmington 562
Cambridge 506
Hong Kong 440
Ann Arbor 391
Dearborn 378
Dublin 292
Princeton 280
Nyköping 279
Izmir 224
Dong Ket 211
The Dalles 193
Boardman 187
Beijing 184
Chicago 157
Rome 133
Lauterbourg 127
Los Angeles 122
San Mateo 109
Ho Chi Minh City 105
San Diego 97
New York 82
Como 76
Hanoi 75
London 74
Santa Clara 68
Council Bluffs 67
Tokyo 66
Munich 63
Orem 57
Ogden 55
Kocaeli 50
São Paulo 49
Mexico City 41
Guangzhou 34
Kunming 33
Düsseldorf 32
Hefei 32
Turku 32
Washington 32
Chennai 31
Des Moines 31
Buffalo 30
Montreal 29
Manchester 28
Verona 28
Atlanta 27
Warsaw 27
Phoenix 25
Johannesburg 24
Boston 22
Shanghai 22
Denver 21
Mumbai 21
Stockholm 21
Brooklyn 19
Nanjing 19
Frankfurt am Main 18
Nanchang 18
Toronto 18
Hangzhou 17
Helsinki 17
Brussels 16
Norwalk 16
Paris 16
Abuja 15
Da Nang 15
Varese 15
Amsterdam 14
Brno 13
Clausthal-Zellerfeld 13
Fuzhou 13
Jinan 13
Nuremberg 13
San Francisco 13
Shenzhen 13
Berlin 12
Elk Grove Village 12
Poplar 12
Rio de Janeiro 12
West Jordan 12
Kilburn 11
Vienna 11
Baghdad 10
Bari 10
Campinas 10
New Delhi 10
Philadelphia 10
Changsha 9
Chiswick 9
Totale 18.493
Nome #
1,3-Dipolar cycloadditions to nitrogen-substituted allenes 1.198
1,3-Dipolar cycloadditions to allenes 1.144
C-C, C-O, C-N Bond Formation on sp2-Carbon by Pd(II)-Catalyzed Reactions Involving Oxidant Agents 261
Boehmeriasin A as new lead compound for the inhibition of topoisomerases and SIRT2 252
Copper(II)-catalyzed alkoxyhalogenation of alkynyl ureas and amides as a route to haloalkylidene substituted heterocycles 220
A facile synthesis of flumazenil analogues 220
(Diacyloxyiodo)benzenes-Driven Palladium-Catalyzed Cyclizations of Unsaturated N-Sulfonylamides: Opportunities of Path Selection 219
A synthetic route to [1,2,4]triazolo[1,5-a][4,1]benzoxazepines 212
Intramolecular Oxidative Palladium-Catalyzed Amination Involving Double C-H Functionalization of Unactivated Olefins 211
A New Entry to [1,2,4]Triazolo[1,5-a][1,4]benzodiazepin-6-ones via Intramolecular Nitrilimine Cycloaddition to the Cyano Group 210
Stereoselective intramolecular cycloadditions of homochiral nitrile imines: synthesis of enantiomerically pure 3,3a-dihydro-pyrazolo[1,5-a][1,4] benzodiazepine-6(4H)-ones 210
Synthesis and biological evaluation of 1,7,8,8a-tetrahydro-3H-oxazolo[3,4-a]pyrazin-6(5H)-ones as antitumoral agents 209
An alternative synthesis of 2-alkylidene-3,4-dihydro-2H-1,4-benzoxazines by intramolecular gold-catalyzed hydroalkoxylation of 2-(prop-2-yn-1-ylamino)-phenols 206
Palladium-catalyzed domino carbopalladation/5-exo-allylic amination of α-amino allenamides: an efficient entry to enantiopure imidazolidinones 201
Synthesis of Pironetin-Dumetorine Hybrids as Tubulin Binders 201
Access to pyrrolo-pyridines by gold-catalyzed hydroarylation of pyrroles tethered to terminal alkynes 199
Dipolarophilic behavior of the isoxazole ring in intramolecular nitrilimine cycloadditions 198
Ruthenium-Catalyzed Hydroamination of Aminoallenes: an Approach to Vinyl Substituted Heterocycles 195
A valuable approach to enantiopure partially saturated pyrrolo- and indolo[1,2-a]indoles by intramolecular nitrone cycloadditions to the cyclohexene ring 192
Synthesis of 1,4-benzodiazepinones via palladium-catalysed allene carbopalladation/amination domino sequence 192
Intra-Intermolecular Palladium-Catalyzed Domino Reactions of Glycine Allylamides for the Synthesis of Diversely Functionalized Piperazinones 190
SYNTHESIS OF ENANTIOPURE 4-AMINO-3-HYDROXYMETHYL-TETRAHYDROQUINOLINES VIA AN INTRAMOLECULAR NITRONE CYCLOADDITION 188
Selective intramolecular palladium(II)-catalyzed aminooxygenation vs. diamination of alkenylureas: efficient microwave-assisted reactions to bicyclic piperazinones 186
5-Heterosubstituted 4-methylene-4,5-dihydroisoxazoles: Ready accessibility and versatile reactivity 185
Palladium-Catalysed Carbo- and Hydroamination of Allenyl Ethers and Aminoallenes: Available Entry to Nitrogen-Containing Benzo-Fused Rings 184
Palladium(II)/copper halide/solvent combination for selective intramolecular domino reactions of indole carboxylic acid allylamides. An unprecedented arylation/esterification sequence 182
New Mechanistic Evidence on the Reaction between Sulfonylallenes and Nitrile Oxides 181
Solvent- and ligand-free palladium-catalyzed amination of aryl halides 181
Efficient Approach to the Unknown Isoxazolo[3,4-d]thieno[2,3-b]pyridine System by Regioselective Intramolecular Nitrone Cycloadditions 178
Recent advances in heterobimetallic palladium(ii)/copper(ii) catalyzed domino difunctionalization of carbon–carbon multiple bonds 178
Synthesis of enantiopure 3-hydroxymethylchromanes via intramolecular nitrone cycloaddition 177
Intramolecular oxidative palladium-catalyzed diamination reactions of alkenyl sulfamates: an efficient synthesis of [1,2,5]thiadiazolo-fused piperazinones 177
The intramolecular azide cycloaddition route to triazolam analogues 176
A valuable heterocyclic ring transformation: from isoxazolin-5(2H)-ones to quinolines 175
Transition metal complexation in 1,3-dipolar cycloadditions 174
Diastereoselective synthesis of bis(3,5)pyrazolophanes by sequential inter- and intramolecular cycloadditions of homochiral nitrilimines 173
N,N-Disubstituted Propargylamines as Tools in the Sequential 1,3-Dipolar Cycloaddition/Arylation Processes to the Formation of Polyheterocyclic Systems 173
Intramolecular azide cycloadditions leading to [1,2,3]triazolo[1,5-a]quinoxalines 173
Transition metal-catalyzed hydroamination and carboamination reactions of anthranilic allenamides as a route to 2-vinyl- and 2-(a-styryl)-quinazolin-4-one derivatives 172
Dehydrogenative Allylic Aminations of But-3-enoic Acid Derivatives 172
Palladium-Catalyzed dual C-H or N-H functionalization of unfunctionalized indole derivatives with alkenes and arenes 171
Pyrrolizidine and indolizidine syntheses involving 1,3-dipolar cycloadditions 170
Intramolecular oxidative Pd(II)-catalyzed alkoxylation of 3-aza-5-alkenols with O2 as sole oxidant: mild conditions for the synthesis of 1,4-oxazine derivatives 170
Intramolecular Aminoazidation of Unactivated Terminal Alkenes by Palladium-Catalyzed Reactions with Hydrogen Peroxide as the Oxidant 170
A new synthesis of flumazenil suitable for fluorine-18 labeling 169
Synthesis of Bis-(3,5)pyrazolophanes by Sequential Intermolecular-Intramolecular Nitrilimine Cycloadditions 168
Thermal behaviour of dipolarophile-containing acyl azides: intramolecular cycloaddition versus Curtius rearrangement 168
New Access to Kainic Acid via Intramolecular Palladium-Catalyzed Allylic Alkylation 167
Intramolecular Cycloadditions of Nitrones Derived from 1-Allyl-2-pyrrolecarbaldehyde as a Route to Racemic and Enantiopure Pyrrolizidines and Indolizidines 165
Uncommon intramolecular palladium-catalyzed cyclization of indole derivatives 165
Chimica degli eterocicli 165
The first case of asymmetric induction in intramolecular nitrile imine cycloadditions: synthesis of enantiopure 3-substituted 6-oxo-2,3,3a,5-tetrahydro-4-carbomethoxy-furo[3,4-c]pyrazoles 164
L-alanine benzylester as chiral inductor: Synthesis of enantiopure pyrazolo[1,5-a]-[1,4]benzodiazepine-4-ones via intramolecular nitrilimine cycloadditions 164
Enantiopure 2-piperidylacetaldehyde as useful building block in the diversity-oriented synthesis of polycyclic piperidine derivatives 164
A new protocol for the conversion of isoxazolidines to 1,3-aminoalcohols 164
Regiochemical aspects of intramolecular cycloadditions of nitrones derived from N-(2-alkenyl)-2-pyrrolecarbaldehydes. Competitive entries to pyrrolizidine and indolizidine derivatives 163
Palladium-catalyzed C-N bond formation via direct C-H bond functionalization. Recent developments in heterocyclic synthesis 163
Stereoselective intramolecular cycloadditions of homochiral N-alkenoyl aryl azides 162
Regioselective Intramolecular Cycloaddition of C-(1-Acryloyl-2-pyrrolyl)-N-benzylnitrone: Entry to 6-Hydroxy-5-oxoindolizidines 162
Synthetic approach to imidazo[1,2-a]pyridine derivatives by the intramolecular nitrone cycloaddition methodology 162
Intramolecular Pd(II)-Catalyzed Cyclization of Propargylamides: Straightforward Synthesis of 5-Oxazole-carbaldehydes 162
Palladium-Catalyzed Cyclization/Carbonylation as a Direct Route to 4-[(Methoxycarbonyl)methyl]-3,4-dihydroisoquinolinones 162
Pd-Catalyzed Intramolecular Cyclization of Pyrrolo-2-carboxamides: Regiodivergent Routes to Pyrrolo-pyrazines and Pyrrolo-pyridines 160
A Valuable Synthesis of Pyrrolo[1,2-a]quinoxalines, Indolo[1,2-a]quinoxalines and their Aza-Analogues by Palladium-Catalyzed Intramolecular Carbon-Nitrogen Bond Formation 159
Enantioselective intramolecular nitrone cycloaddition route to 3-(trifluoromethyl)-isoxazolidino[4,3-c]-chroman-4-ones and -quinolin-4-ones 159
Regioselectivity on the palladium-catalyzed intramolecular cyclization of indole derivatives 158
Intramolecular Palladium-Catalyzed Aminocarboxylation of Olefins as a Direct Route to Bicyclic Oxazolidinones 158
Solvent-free, microwave-assisted N-arylation of indolines by using low palladium catalyst loadings 158
Dipolarophilic behaviour of the thiophene ring in intramolecular nitrile imine cycloadditions 157
Selective 7- endo -Cyclization of 3-Aza-5-alkenols through Oxidative Pd(II)-Catalyzed Olefin Oxyarylation 157
Synthesis of enantiopure pyrrolo[3,4-c]pyrazole derivatives via intramolecular cycloaddition of homochiral nitrilimines 156
Dipolarophilic behaviour of (arylsulfonyl)allenes towards nitrilimines 156
Oxidative cleavage of the isoxazolidine ring 154
Synthesis of tetrazolo[1,5-a][1,4]benzodiazepin-6-ones via intramolecular azide cycloadditions onto the cyano group 154
Nitrilimine cycloadditions onto partially saturated furo[3,4-c]thieno[2,3-d]pyrazoles. A problem in site selectivity 153
Access to pyrralo- and pyrido[1,2-a]indole derivatives by intramolecular nitrone cycloadditions. Effect of steric factors on the regioselective product formation 151
Iodoamination of Alkenyl Sulfonamides by Potassium Iodide and Hydrogen Peroxide in Aqueous Medium 151
Palladium-mediated Approach to Dibenzo[b,e][1,4]diazepines and Benzopyrido-analogues. An Efficient Synthesis of Tarpane 150
Access to a Novel Class of Tetracyclic 1,4-Benzodiazepin-5-ones Starting from alpha-Aminoacids by Pd-Catalyzed Amination/1,3-Dipolar Cycloaddition as Key Steps 150
Synthesis of pyrazolo[1,5-a]quinoxalines 150
A facile synthesis of 2-methyl-1,4-benzodiazepin-5-ones via intramolecular azide cycloaddition 149
Nitrilimine cycloadditions in aqueous media 148
Intramolecular nitrile imide cycloadditions onto the furan ring: synthesis of the new 3a,4-dihydro-6H-difuro[3,2-c;3,4-d]pyrazole skeleton 148
Direct Synthesis of Fluorescent Oxazolo-phenoxazines by Copper-Catalyzed/Hypervalent Iodine(III)-Mediated Dimerization/Cyclization of 2-Benzylamino-phenols 147
Relative and absolute stereocontrol in intramolecular nitrone cycloadditions to the cyclohexene ring 146
Asymmetric induction by the (S)-1-phenylethyl group in intramolecular nitrile imine cycloadditions giving enantiopure 3,3a-dihydro-pyrazolo[1,5-alpha][1,4]benzodiazepine-4(6H)-ones 145
Synthesis of enantiopure 4-amino-6-fluoro-3-(hydroxymethyl)chromanes via intramolecular nitrone cycloadditions 145
Intramolecular cycloadditions of nitrones derived from optically active 1-alkenyl-2-imidazolecarbaldehydes: regio- and diastereoselectivity 144
Synthesis and Biological Evaluation of Migrastatin Macrotriazoles 144
Intramolecular cycloadditions of N-alkenoyl aryl azides 143
Intramolecular Azide Cycloaddition en Route to the New Pyrrolo[2,1-c][1,2,3]triazolo[1,5-a][1,4]benzodiazepine Skeleton 143
Efficient Synthesis of N-Methoxyindoles via Alkylative Cycloaddition of Nitrosoarenes with Alkynes 143
Synthesis of N-(5-amino-2-pyrimidyl)-N '-[4-(p-fluorophenyl)-4-oxobutyl]piperazine, a useful intermediate to antipsychotic agents 142
Synthesis of 5-hydroxymethyl-1,4-dioxan-2-one 141
Copper-Catalyzed Alkoxylation as Key Step to Convert Isatin to Oxazinoindol-2-one Derivatives 141
Divergent Palladium- and Platinum-Catalyzed Intramolecular Hydroamination/Hydroarylation of O-Propargyl-2-aminophenols 141
Diastereoselective nitrilimine cycloaddition to the C = N bond of enantiopure 1,4-benzodiazepinones 140
Entry to nitrogen-containing heterocycles by base-promoted heterocyclization on allenylamides of L-a-aminoacids 140
Transition metal catalyzed azidation reactions 140
Novel aspects of the silver carbonate promoted reaction of hydrazonyl chlorides with homoallylic and homopropargylic alcohols 139
Totale 19.025
Categoria #
all - tutte 92.439
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 92.439


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021713 0 0 0 0 0 0 0 0 0 181 203 329
2021/20221.507 172 316 115 34 32 46 139 56 73 198 152 174
2022/20231.883 230 89 135 186 138 412 14 272 226 53 75 53
2023/20243.001 422 400 462 598 628 188 34 57 89 28 27 68
2024/20252.165 52 39 446 47 62 112 61 127 229 142 188 660
2025/20266.878 414 689 1.460 887 648 369 1.176 394 545 296 0 0
Totale 25.039