BROGGINI, GIANLUIGI
 Distribuzione geografica
Continente #
NA - Nord America 9.407
EU - Europa 5.172
AS - Asia 1.189
Continente sconosciuto - Info sul continente non disponibili 16
SA - Sud America 9
OC - Oceania 5
AF - Africa 2
Totale 15.800
Nazione #
US - Stati Uniti d'America 9.393
IT - Italia 2.458
UA - Ucraina 1.012
TR - Turchia 507
SE - Svezia 452
VN - Vietnam 330
IE - Irlanda 291
CN - Cina 279
DE - Germania 259
FI - Finlandia 249
GB - Regno Unito 244
FR - Francia 58
JP - Giappone 38
ES - Italia 21
BE - Belgio 18
CH - Svizzera 17
IN - India 17
EU - Europa 16
CZ - Repubblica Ceca 15
RU - Federazione Russa 15
NL - Olanda 13
CA - Canada 12
AT - Austria 10
BR - Brasile 8
PT - Portogallo 7
RO - Romania 7
NO - Norvegia 6
AU - Australia 5
SG - Singapore 4
BG - Bulgaria 3
DK - Danimarca 3
GR - Grecia 3
PL - Polonia 3
ID - Indonesia 2
IL - Israele 2
MY - Malesia 2
PA - Panama 2
AE - Emirati Arabi Uniti 1
AL - Albania 1
AZ - Azerbaigian 1
BD - Bangladesh 1
BO - Bolivia 1
BT - Bhutan 1
BY - Bielorussia 1
DZ - Algeria 1
ET - Etiopia 1
HU - Ungheria 1
KZ - Kazakistan 1
LU - Lussemburgo 1
MD - Moldavia 1
ME - Montenegro 1
MM - Myanmar 1
MO - Macao, regione amministrativa speciale della Cina 1
SI - Slovenia 1
SK - Slovacchia (Repubblica Slovacca) 1
TH - Thailandia 1
Totale 15.800
Città #
Milan 1.723
Fairfield 1.649
Woodbridge 927
Jacksonville 780
Ashburn 764
Houston 667
Seattle 659
Chandler 628
Wilmington 560
Cambridge 506
Ann Arbor 391
Dearborn 378
Dublin 291
Princeton 280
Nyköping 279
Izmir 224
Dong Ket 211
Rome 130
San Mateo 109
San Diego 97
Como 71
Ogden 55
Kocaeli 50
Beijing 46
London 39
Tokyo 36
Boardman 34
Kunming 33
Washington 32
Düsseldorf 31
Hefei 31
Verona 28
Nanjing 18
Nanchang 17
New York 16
Norwalk 16
Brussels 15
Los Angeles 15
Brno 13
Clausthal-Zellerfeld 13
Berlin 12
Fuzhou 12
Jinan 12
West Jordan 12
Chicago 11
Guangzhou 11
Kilburn 11
Bari 9
Chiswick 9
Frankfurt am Main 9
Hounslow 9
Paris 9
Toronto 9
Vienna 9
Auburn Hills 8
Edinburgh 8
Munich 8
New Bedfont 8
Prescot 7
Shanghai 7
Florence 6
Islington 6
Lisbon 6
Oslo 6
São Paulo 6
Timisoara 6
Acton 5
Amsterdam 5
Besana In Brianza 5
Brescia 5
Changsha 5
Giussano 5
Perugia 5
Phoenix 5
Rozzano 5
San Francisco 5
Shenyang 5
Southwark 5
Wandsworth 5
Wuhan 5
Bristol 4
Chengdu 4
Hebei 4
Helsinki 4
Lappeenranta 4
Madrid 4
Mumbai 4
Naples 4
Philadelphia 4
Redmond 4
Rouen 4
Stockholm 4
Zhengzhou 4
Athens 3
Brugherio 3
Busto Arsizio 3
Canberra 3
Gaggiano 3
Magenta 3
Manchester 3
Totale 12.231
Nome #
1,3-Dipolar cycloadditions to nitrogen-substituted allenes 252
1,3-Dipolar cycloadditions to allenes 186
Boehmeriasin A as new lead compound for the inhibition of topoisomerases and SIRT2 186
C-C, C-O, C-N Bond Formation on sp2-Carbon by Pd(II)-Catalyzed Reactions Involving Oxidant Agents 185
Copper(II)-catalyzed alkoxyhalogenation of alkynyl ureas and amides as a route to haloalkylidene substituted heterocycles 172
Palladium-catalyzed domino carbopalladation/5-exo-allylic amination of α-amino allenamides: an efficient entry to enantiopure imidazolidinones 169
Synthesis and biological evaluation of 1,7,8,8a-tetrahydro-3H-oxazolo[3,4-a]pyrazin-6(5H)-ones as antitumoral agents 169
Stereoselective intramolecular cycloadditions of homochiral nitrile imines: synthesis of enantiomerically pure 3,3a-dihydro-pyrazolo[1,5-a][1,4] benzodiazepine-6(4H)-ones 167
Synthesis of Pironetin-Dumetorine Hybrids as Tubulin Binders 163
(Diacyloxyiodo)benzenes-Driven Palladium-Catalyzed Cyclizations of Unsaturated N-Sulfonylamides: Opportunities of Path Selection 162
Selective intramolecular palladium(II)-catalyzed aminooxygenation vs. diamination of alkenylureas: efficient microwave-assisted reactions to bicyclic piperazinones 158
A facile synthesis of flumazenil analogues 157
An alternative synthesis of 2-alkylidene-3,4-dihydro-2H-1,4-benzoxazines by intramolecular gold-catalyzed hydroalkoxylation of 2-(prop-2-yn-1-ylamino)-phenols 155
Solvent- and ligand-free palladium-catalyzed amination of aryl halides 152
SYNTHESIS OF ENANTIOPURE 4-AMINO-3-HYDROXYMETHYL-TETRAHYDROQUINOLINES VIA AN INTRAMOLECULAR NITRONE CYCLOADDITION 151
Ruthenium-Catalyzed Hydroamination of Aminoallenes: an Approach to Vinyl Substituted Heterocycles 151
Intramolecular Oxidative Palladium-Catalyzed Amination Involving Double C-H Functionalization of Unactivated Olefins 151
Intra-Intermolecular Palladium-Catalyzed Domino Reactions of Glycine Allylamides for the Synthesis of Diversely Functionalized Piperazinones 150
Synthesis of 1,4-benzodiazepinones via palladium-catalysed allene carbopalladation/amination domino sequence 149
A synthetic route to [1,2,4]triazolo[1,5-a][4,1]benzoxazepines 148
A New Entry to [1,2,4]Triazolo[1,5-a][1,4]benzodiazepin-6-ones via Intramolecular Nitrilimine Cycloaddition to the Cyano Group 147
Transition metal complexation in 1,3-dipolar cycloadditions 145
New Mechanistic Evidence on the Reaction between Sulfonylallenes and Nitrile Oxides 144
Palladium(II)/copper halide/solvent combination for selective intramolecular domino reactions of indole carboxylic acid allylamides. An unprecedented arylation/esterification sequence 143
The intramolecular azide cycloaddition route to triazolam analogues 142
Intramolecular azide cycloadditions leading to [1,2,3]triazolo[1,5-a]quinoxalines 142
Access to pyrrolo-pyridines by gold-catalyzed hydroarylation of pyrroles tethered to terminal alkynes 141
Dehydrogenative Allylic Aminations of But-3-enoic Acid Derivatives 141
New Access to Kainic Acid via Intramolecular Palladium-Catalyzed Allylic Alkylation 138
Recent advances in heterobimetallic palladium(ii)/copper(ii) catalyzed domino difunctionalization of carbon–carbon multiple bonds 136
Synthesis of enantiopure 3-hydroxymethylchromanes via intramolecular nitrone cycloaddition 135
Palladium-Catalysed Carbo- and Hydroamination of Allenyl Ethers and Aminoallenes: Available Entry to Nitrogen-Containing Benzo-Fused Rings 135
Synthesis of Bis-(3,5)pyrazolophanes by Sequential Intermolecular-Intramolecular Nitrilimine Cycloadditions 134
Diastereoselective synthesis of bis(3,5)pyrazolophanes by sequential inter- and intramolecular cycloadditions of homochiral nitrilimines 134
N,N-Disubstituted Propargylamines as Tools in the Sequential 1,3-Dipolar Cycloaddition/Arylation Processes to the Formation of Polyheterocyclic Systems 134
Palladium-Catalyzed Cyclization/Carbonylation as a Direct Route to 4-[(Methoxycarbonyl)methyl]-3,4-dihydroisoquinolinones 133
5-Heterosubstituted 4-methylene-4,5-dihydroisoxazoles: Ready accessibility and versatile reactivity 132
Thermal behaviour of dipolarophile-containing acyl azides: intramolecular cycloaddition versus Curtius rearrangement 132
Intramolecular oxidative palladium-catalyzed diamination reactions of alkenyl sulfamates: an efficient synthesis of [1,2,5]thiadiazolo-fused piperazinones 132
Solvent-free, microwave-assisted N-arylation of indolines by using low palladium catalyst loadings 129
The first case of asymmetric induction in intramolecular nitrile imine cycloadditions: synthesis of enantiopure 3-substituted 6-oxo-2,3,3a,5-tetrahydro-4-carbomethoxy-furo[3,4-c]pyrazoles 128
Regiochemical aspects of intramolecular cycloadditions of nitrones derived from N-(2-alkenyl)-2-pyrrolecarbaldehydes. Competitive entries to pyrrolizidine and indolizidine derivatives 128
Intramolecular Palladium-Catalyzed Aminocarboxylation of Olefins as a Direct Route to Bicyclic Oxazolidinones 128
Transition metal-catalyzed hydroamination and carboamination reactions of anthranilic allenamides as a route to 2-vinyl- and 2-(a-styryl)-quinazolin-4-one derivatives 128
Pyrrolizidine and indolizidine syntheses involving 1,3-dipolar cycloadditions 127
Palladium-Catalyzed dual C-H or N-H functionalization of unfunctionalized indole derivatives with alkenes and arenes 127
Intramolecular Cycloadditions of Nitrones Derived from 1-Allyl-2-pyrrolecarbaldehyde as a Route to Racemic and Enantiopure Pyrrolizidines and Indolizidines 126
Synthetic approach to imidazo[1,2-a]pyridine derivatives by the intramolecular nitrone cycloaddition methodology 126
Efficient Approach to the Unknown Isoxazolo[3,4-d]thieno[2,3-b]pyridine System by Regioselective Intramolecular Nitrone Cycloadditions 126
Uncommon intramolecular palladium-catalyzed cyclization of indole derivatives 125
Stereoselective intramolecular cycloadditions of homochiral N-alkenoyl aryl azides 125
Dipolarophilic behavior of the isoxazole ring in intramolecular nitrilimine cycloadditions 125
Intramolecular oxidative Pd(II)-catalyzed alkoxylation of 3-aza-5-alkenols with O2 as sole oxidant: mild conditions for the synthesis of 1,4-oxazine derivatives 125
A valuable approach to enantiopure partially saturated pyrrolo- and indolo[1,2-a]indoles by intramolecular nitrone cycloadditions to the cyclohexene ring 124
Dipolarophilic behaviour of (arylsulfonyl)allenes towards nitrilimines 124
Pd-Catalyzed Intramolecular Cyclization of Pyrrolo-2-carboxamides: Regiodivergent Routes to Pyrrolo-pyrazines and Pyrrolo-pyridines 123
Palladium-mediated Approach to Dibenzo[b,e][1,4]diazepines and Benzopyrido-analogues. An Efficient Synthesis of Tarpane 123
L-alanine benzylester as chiral inductor: Synthesis of enantiopure pyrazolo[1,5-a]-[1,4]benzodiazepine-4-ones via intramolecular nitrilimine cycloadditions 122
Intramolecular Pd(II)-Catalyzed Cyclization of Propargylamides: Straightforward Synthesis of 5-Oxazole-carbaldehydes 121
Palladium-catalyzed C-N bond formation via direct C-H bond functionalization. Recent developments in heterocyclic synthesis 121
Enantiopure 2-piperidylacetaldehyde as useful building block in the diversity-oriented synthesis of polycyclic piperidine derivatives 121
Regioselective Intramolecular Cycloaddition of C-(1-Acryloyl-2-pyrrolyl)-N-benzylnitrone: Entry to 6-Hydroxy-5-oxoindolizidines 120
Synthesis of enantiopure pyrrolo[3,4-c]pyrazole derivatives via intramolecular cycloaddition of homochiral nitrilimines 119
A valuable heterocyclic ring transformation: from isoxazolin-5(2H)-ones to quinolines 119
Synthesis of tetrazolo[1,5-a][1,4]benzodiazepin-6-ones via intramolecular azide cycloadditions onto the cyano group 119
Regioselectivity on the palladium-catalyzed intramolecular cyclization of indole derivatives 118
Synthesis of enantiopure 4-amino-6-fluoro-3-(hydroxymethyl)chromanes via intramolecular nitrone cycloadditions 118
Synthesis and Biological Evaluation of Migrastatin Macrotriazoles 116
Nitrilimine cycloadditions onto partially saturated furo[3,4-c]thieno[2,3-d]pyrazoles. A problem in site selectivity 114
Relative and absolute stereocontrol in intramolecular nitrone cycloadditions to the cyclohexene ring 114
Intramolecular cycloadditions of N-alkenoyl aryl azides 113
Diastereoselective nitrilimine cycloaddition to the C = N bond of enantiopure 1,4-benzodiazepinones 113
A new protocol for the conversion of isoxazolidines to 1,3-aminoalcohols 113
Divergent Palladium- and Platinum-Catalyzed Intramolecular Hydroamination/Hydroarylation of O-Propargyl-2-aminophenols 113
Intramolecular nitrile imide cycloadditions onto the furan ring: synthesis of the new 3a,4-dihydro-6H-difuro[3,2-c;3,4-d]pyrazole skeleton 112
Intramolecular Aminoazidation of Unactivated Terminal Alkenes by Palladium-Catalyzed Reactions with Hydrogen Peroxide as the Oxidant 112
Intramolecular Azide Cycloaddition en Route to the New Pyrrolo[2,1-c][1,2,3]triazolo[1,5-a][1,4]benzodiazepine Skeleton 111
Efficient Synthesis of N-Methoxyindoles via Alkylative Cycloaddition of Nitrosoarenes with Alkynes 111
Synthesis of pyrazolo[1,5-a]quinoxalines 111
Copper-Catalyzed Alkoxylation as Key Step to Convert Isatin to Oxazinoindol-2-one Derivatives 111
Microwave-Assisted Intramolecular Cyclization of Electron-Rich HeterocycleDerivatives by a Palladium-Catalyzed Coupling Reaction 110
A new synthesis of flumazenil suitable for fluorine-18 labeling 109
Tunable Pd-Catalyzed Cyclization of Indole-2-carboxylic Acid Allenamides: Carboamination vs Microwave-Assisted Hydroamination 108
Selective 7- endo -Cyclization of 3-Aza-5-alkenols through Oxidative Pd(II)-Catalyzed Olefin Oxyarylation 108
Nitrilimine cycloadditions in aqueous media 107
Intramolecular cycloadditions of nitrones derived from optically active 1-alkenyl-2-imidazolecarbaldehydes: regio- and diastereoselectivity 107
Enantioselective intramolecular nitrone cycloaddition route to 3-(trifluoromethyl)-isoxazolidino[4,3-c]-chroman-4-ones and -quinolin-4-ones 106
Novel aspects of the silver carbonate promoted reaction of hydrazonyl chlorides with homoallylic and homopropargylic alcohols 105
Synthesis of 5-hydroxymethyl-1,4-dioxan-2-one 105
Oxidative cleavage of the isoxazolidine ring 104
Dipolarophilic behaviour of the thiophene ring in intramolecular nitrile imine cycloadditions 104
Synthesis and biological evaluation of pyrimidine-oxazolidin-2-arylimino hybrid molecules as antibacterial agents 104
Chimica degli eterocicli 102
Effective Synthesis of Enantiopure [1,2,3]Triazolo[1,5-a]- and Pyrazolo[1,5-a]-pyrrolo[2,1-c][1,4]benzodiazepines by Diastereoselective Intramolecular Azide and Nitrilimine Cycloadditions 102
A Valuable Synthesis of Pyrrolo[1,2-a]quinoxalines, Indolo[1,2-a]quinoxalines and their Aza-Analogues by Palladium-Catalyzed Intramolecular Carbon-Nitrogen Bond Formation 102
Pd-Catalyzed Cyclization of 1-Allyl-2-indolecarboxamides by Intramolecular Amidation of Unactivated Ethylenic Bond 102
Synthesis of N-(5-amino-2-pyrimidyl)-N '-[4-(p-fluorophenyl)-4-oxobutyl]piperazine, a useful intermediate to antipsychotic agents 98
Efficient palladium-catalyzed direct arylation of azines and diazines using ligand-free conditions 98
Synthesis of pyrazole-containing azacrown ethers by intramolecular nitrilimine cycloadditions 98
Access to pyrralo- and pyrido[1,2-a]indole derivatives by intramolecular nitrone cycloadditions. Effect of steric factors on the regioselective product formation 95
Totale 12.956
Categoria #
all - tutte 58.272
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 58.272


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/20203.711 185 153 199 737 252 463 500 424 281 242 62 213
2020/20212.423 56 233 106 228 130 262 162 203 330 181 203 329
2021/20221.507 172 316 115 34 32 46 139 56 73 198 152 174
2022/20231.883 230 89 135 186 138 412 14 272 226 53 75 53
2023/20243.001 422 400 462 598 628 188 34 57 89 28 27 68
2024/202538 38 0 0 0 0 0 0 0 0 0 0 0
Totale 16.034