BROGGINI, GIANLUIGI
 Distribuzione geografica
Continente #
NA - Nord America 14.701
EU - Europa 6.076
AS - Asia 4.264
SA - Sud America 437
Continente sconosciuto - Info sul continente non disponibili 265
AF - Africa 73
OC - Oceania 6
Totale 25.822
Nazione #
US - Stati Uniti d'America 14.517
IT - Italia 2.629
SG - Singapore 1.375
UA - Ucraina 1.021
CN - Cina 937
VN - Vietnam 637
TR - Turchia 522
SE - Svezia 516
HK - Hong Kong 454
BR - Brasile 360
GB - Regno Unito 359
DE - Germania 352
FI - Finlandia 297
IE - Irlanda 292
FR - Francia 205
RU - Federazione Russa 173
IN - India 99
CA - Canada 87
JP - Giappone 72
MX - Messico 70
ES - Italia 52
BD - Bangladesh 41
PL - Polonia 33
ZA - Sudafrica 31
IQ - Iraq 27
NL - Olanda 25
AR - Argentina 24
BE - Belgio 19
CH - Svizzera 17
EU - Europa 16
CZ - Repubblica Ceca 15
NG - Nigeria 15
AT - Austria 13
VE - Venezuela 13
ID - Indonesia 12
AE - Emirati Arabi Uniti 10
EC - Ecuador 9
PK - Pakistan 9
LT - Lituania 8
PT - Portogallo 8
SA - Arabia Saudita 8
MD - Moldavia 7
RO - Romania 7
TN - Tunisia 7
AU - Australia 6
CL - Cile 6
CO - Colombia 6
NO - Norvegia 6
NP - Nepal 6
PE - Perù 6
IL - Israele 5
MY - Malesia 5
PH - Filippine 5
PY - Paraguay 5
UZ - Uzbekistan 5
AZ - Azerbaigian 4
BG - Bulgaria 4
GR - Grecia 4
JO - Giordania 4
TH - Thailandia 4
TW - Taiwan 4
UY - Uruguay 4
BB - Barbados 3
BO - Bolivia 3
DK - Danimarca 3
EG - Egitto 3
GT - Guatemala 3
HN - Honduras 3
KE - Kenya 3
KZ - Kazakistan 3
MA - Marocco 3
PA - Panama 3
ZW - Zimbabwe 3
AL - Albania 2
BN - Brunei Darussalam 2
CR - Costa Rica 2
DM - Dominica 2
DZ - Algeria 2
GP - Guadalupe 2
HU - Ungheria 2
JM - Giamaica 2
LB - Libano 2
OM - Oman 2
PS - Palestinian Territory 2
SN - Senegal 2
SV - El Salvador 2
TT - Trinidad e Tobago 2
BH - Bahrain 1
BT - Bhutan 1
BY - Bielorussia 1
CI - Costa d'Avorio 1
DO - Repubblica Dominicana 1
ET - Etiopia 1
GA - Gabon 1
GD - Grenada 1
GY - Guiana 1
HR - Croazia 1
IR - Iran 1
KG - Kirghizistan 1
LU - Lussemburgo 1
Totale 25.563
Città #
Dallas 1.909
Milan 1.756
Fairfield 1.649
Ashburn 1.112
San Jose 929
Woodbridge 927
Singapore 808
Jacksonville 781
Houston 685
Seattle 670
Chandler 628
Wilmington 562
Cambridge 506
Hong Kong 447
Ann Arbor 391
Dearborn 379
Dublin 293
Princeton 280
Nyköping 279
Izmir 224
Dong Ket 211
Beijing 197
The Dalles 194
Boardman 187
Chicago 159
Rome 136
Los Angeles 130
Council Bluffs 128
Lauterbourg 127
San Mateo 109
Ho Chi Minh City 105
San Diego 98
Santa Clara 98
New York 91
Como 76
Hanoi 76
London 74
Tokyo 66
Munich 63
Orem 58
Ogden 55
Kocaeli 50
São Paulo 49
Mexico City 45
Guangzhou 34
Kunming 33
Buffalo 32
Düsseldorf 32
Hefei 32
Turku 32
Washington 32
Chennai 31
Des Moines 31
Atlanta 30
Montreal 30
Verona 29
Manchester 28
Shanghai 28
Warsaw 27
Phoenix 25
Johannesburg 24
Boston 22
Denver 22
Brooklyn 21
Mumbai 21
Stockholm 21
Toronto 20
Varese 20
Nanjing 19
Frankfurt am Main 18
Nanchang 18
Hangzhou 17
Helsinki 17
Paris 17
Brussels 16
Norwalk 16
Abuja 15
Da Nang 15
San Francisco 15
Amsterdam 14
Brno 13
Clausthal-Zellerfeld 13
Fuzhou 13
Jinan 13
Nuremberg 13
Philadelphia 13
Shenzhen 13
Berlin 12
Elk Grove Village 12
Poplar 12
Rio de Janeiro 12
West Jordan 12
Kilburn 11
Las Vegas 11
Vienna 11
Baghdad 10
Bari 10
Campinas 10
Changsha 10
New Delhi 10
Totale 18.885
Nome #
1,3-Dipolar cycloadditions to nitrogen-substituted allenes 1.207
1,3-Dipolar cycloadditions to allenes 1.151
C-C, C-O, C-N Bond Formation on sp2-Carbon by Pd(II)-Catalyzed Reactions Involving Oxidant Agents 272
Palladium-catalyzed domino carbopalladation/5-exo-allylic amination of α-amino allenamides: an efficient entry to enantiopure imidazolidinones 264
Boehmeriasin A as new lead compound for the inhibition of topoisomerases and SIRT2 258
Dipolarophilic behavior of the isoxazole ring in intramolecular nitrilimine cycloadditions 240
Copper(II)-catalyzed alkoxyhalogenation of alkynyl ureas and amides as a route to haloalkylidene substituted heterocycles 225
A facile synthesis of flumazenil analogues 225
(Diacyloxyiodo)benzenes-Driven Palladium-Catalyzed Cyclizations of Unsaturated N-Sulfonylamides: Opportunities of Path Selection 222
A synthetic route to [1,2,4]triazolo[1,5-a][4,1]benzoxazepines 218
Synthesis and biological evaluation of 1,7,8,8a-tetrahydro-3H-oxazolo[3,4-a]pyrazin-6(5H)-ones as antitumoral agents 215
Synthesis of Pironetin-Dumetorine Hybrids as Tubulin Binders 215
A New Entry to [1,2,4]Triazolo[1,5-a][1,4]benzodiazepin-6-ones via Intramolecular Nitrilimine Cycloaddition to the Cyano Group 213
Intramolecular Oxidative Palladium-Catalyzed Amination Involving Double C-H Functionalization of Unactivated Olefins 213
Stereoselective intramolecular cycloadditions of homochiral nitrile imines: synthesis of enantiomerically pure 3,3a-dihydro-pyrazolo[1,5-a][1,4] benzodiazepine-6(4H)-ones 212
An alternative synthesis of 2-alkylidene-3,4-dihydro-2H-1,4-benzoxazines by intramolecular gold-catalyzed hydroalkoxylation of 2-(prop-2-yn-1-ylamino)-phenols 211
Access to pyrrolo-pyridines by gold-catalyzed hydroarylation of pyrroles tethered to terminal alkynes 201
Synthesis of 1,4-benzodiazepinones via palladium-catalysed allene carbopalladation/amination domino sequence 197
Ruthenium-Catalyzed Hydroamination of Aminoallenes: an Approach to Vinyl Substituted Heterocycles 196
A valuable approach to enantiopure partially saturated pyrrolo- and indolo[1,2-a]indoles by intramolecular nitrone cycloadditions to the cyclohexene ring 195
SYNTHESIS OF ENANTIOPURE 4-AMINO-3-HYDROXYMETHYL-TETRAHYDROQUINOLINES VIA AN INTRAMOLECULAR NITRONE CYCLOADDITION 191
Selective intramolecular palladium(II)-catalyzed aminooxygenation vs. diamination of alkenylureas: efficient microwave-assisted reactions to bicyclic piperazinones 191
Intra-Intermolecular Palladium-Catalyzed Domino Reactions of Glycine Allylamides for the Synthesis of Diversely Functionalized Piperazinones 191
5-Heterosubstituted 4-methylene-4,5-dihydroisoxazoles: Ready accessibility and versatile reactivity 189
Palladium(II)/copper halide/solvent combination for selective intramolecular domino reactions of indole carboxylic acid allylamides. An unprecedented arylation/esterification sequence 188
Palladium-Catalysed Carbo- and Hydroamination of Allenyl Ethers and Aminoallenes: Available Entry to Nitrogen-Containing Benzo-Fused Rings 188
Efficient Approach to the Unknown Isoxazolo[3,4-d]thieno[2,3-b]pyridine System by Regioselective Intramolecular Nitrone Cycloadditions 184
Solvent- and ligand-free palladium-catalyzed amination of aryl halides 183
New Mechanistic Evidence on the Reaction between Sulfonylallenes and Nitrile Oxides 182
The intramolecular azide cycloaddition route to triazolam analogues 182
Intramolecular oxidative palladium-catalyzed diamination reactions of alkenyl sulfamates: an efficient synthesis of [1,2,5]thiadiazolo-fused piperazinones 181
A valuable heterocyclic ring transformation: from isoxazolin-5(2H)-ones to quinolines 180
Recent advances in heterobimetallic palladium(ii)/copper(ii) catalyzed domino difunctionalization of carbon–carbon multiple bonds 180
Synthesis of enantiopure 3-hydroxymethylchromanes via intramolecular nitrone cycloaddition 178
Diastereoselective synthesis of bis(3,5)pyrazolophanes by sequential inter- and intramolecular cycloadditions of homochiral nitrilimines 176
Dehydrogenative Allylic Aminations of But-3-enoic Acid Derivatives 176
N,N-Disubstituted Propargylamines as Tools in the Sequential 1,3-Dipolar Cycloaddition/Arylation Processes to the Formation of Polyheterocyclic Systems 176
Intramolecular azide cycloadditions leading to [1,2,3]triazolo[1,5-a]quinoxalines 176
Transition metal complexation in 1,3-dipolar cycloadditions 176
A new synthesis of flumazenil suitable for fluorine-18 labeling 174
Pyrrolizidine and indolizidine syntheses involving 1,3-dipolar cycloadditions 174
Palladium-Catalyzed dual C-H or N-H functionalization of unfunctionalized indole derivatives with alkenes and arenes 174
New Access to Kainic Acid via Intramolecular Palladium-Catalyzed Allylic Alkylation 173
Transition metal-catalyzed hydroamination and carboamination reactions of anthranilic allenamides as a route to 2-vinyl- and 2-(a-styryl)-quinazolin-4-one derivatives 173
Intramolecular Aminoazidation of Unactivated Terminal Alkenes by Palladium-Catalyzed Reactions with Hydrogen Peroxide as the Oxidant 173
Synthesis of Bis-(3,5)pyrazolophanes by Sequential Intermolecular-Intramolecular Nitrilimine Cycloadditions 172
Intramolecular oxidative Pd(II)-catalyzed alkoxylation of 3-aza-5-alkenols with O2 as sole oxidant: mild conditions for the synthesis of 1,4-oxazine derivatives 172
Thermal behaviour of dipolarophile-containing acyl azides: intramolecular cycloaddition versus Curtius rearrangement 171
Intramolecular Pd(II)-Catalyzed Cyclization of Propargylamides: Straightforward Synthesis of 5-Oxazole-carbaldehydes 170
Palladium-catalyzed C-N bond formation via direct C-H bond functionalization. Recent developments in heterocyclic synthesis 170
Chimica degli eterocicli 169
Intramolecular Cycloadditions of Nitrones Derived from 1-Allyl-2-pyrrolecarbaldehyde as a Route to Racemic and Enantiopure Pyrrolizidines and Indolizidines 168
Uncommon intramolecular palladium-catalyzed cyclization of indole derivatives 167
L-alanine benzylester as chiral inductor: Synthesis of enantiopure pyrazolo[1,5-a]-[1,4]benzodiazepine-4-ones via intramolecular nitrilimine cycloadditions 167
A new protocol for the conversion of isoxazolidines to 1,3-aminoalcohols 167
The first case of asymmetric induction in intramolecular nitrile imine cycloadditions: synthesis of enantiopure 3-substituted 6-oxo-2,3,3a,5-tetrahydro-4-carbomethoxy-furo[3,4-c]pyrazoles 166
Regioselective Intramolecular Cycloaddition of C-(1-Acryloyl-2-pyrrolyl)-N-benzylnitrone: Entry to 6-Hydroxy-5-oxoindolizidines 166
Regiochemical aspects of intramolecular cycloadditions of nitrones derived from N-(2-alkenyl)-2-pyrrolecarbaldehydes. Competitive entries to pyrrolizidine and indolizidine derivatives 166
Palladium-Catalyzed Cyclization/Carbonylation as a Direct Route to 4-[(Methoxycarbonyl)methyl]-3,4-dihydroisoquinolinones 166
Enantiopure 2-piperidylacetaldehyde as useful building block in the diversity-oriented synthesis of polycyclic piperidine derivatives 166
Pd-Catalyzed Intramolecular Cyclization of Pyrrolo-2-carboxamides: Regiodivergent Routes to Pyrrolo-pyrazines and Pyrrolo-pyridines 165
Synthetic approach to imidazo[1,2-a]pyridine derivatives by the intramolecular nitrone cycloaddition methodology 164
A Valuable Synthesis of Pyrrolo[1,2-a]quinoxalines, Indolo[1,2-a]quinoxalines and their Aza-Analogues by Palladium-Catalyzed Intramolecular Carbon-Nitrogen Bond Formation 164
Enantioselective intramolecular nitrone cycloaddition route to 3-(trifluoromethyl)-isoxazolidino[4,3-c]-chroman-4-ones and -quinolin-4-ones 164
Stereoselective intramolecular cycloadditions of homochiral N-alkenoyl aryl azides 163
Intramolecular Palladium-Catalyzed Aminocarboxylation of Olefins as a Direct Route to Bicyclic Oxazolidinones 162
Solvent-free, microwave-assisted N-arylation of indolines by using low palladium catalyst loadings 162
Synthesis of enantiopure pyrrolo[3,4-c]pyrazole derivatives via intramolecular cycloaddition of homochiral nitrilimines 160
Dipolarophilic behaviour of the thiophene ring in intramolecular nitrile imine cycloadditions 160
Nitrilimine cycloadditions onto partially saturated furo[3,4-c]thieno[2,3-d]pyrazoles. A problem in site selectivity 159
Regioselectivity on the palladium-catalyzed intramolecular cyclization of indole derivatives 158
Dipolarophilic behaviour of (arylsulfonyl)allenes towards nitrilimines 158
Selective 7- endo -Cyclization of 3-Aza-5-alkenols through Oxidative Pd(II)-Catalyzed Olefin Oxyarylation 158
Access to pyrralo- and pyrido[1,2-a]indole derivatives by intramolecular nitrone cycloadditions. Effect of steric factors on the regioselective product formation 157
Direct Synthesis of Fluorescent Oxazolo-phenoxazines by Copper-Catalyzed/Hypervalent Iodine(III)-Mediated Dimerization/Cyclization of 2-Benzylamino-phenols 157
Synthesis of tetrazolo[1,5-a][1,4]benzodiazepin-6-ones via intramolecular azide cycloadditions onto the cyano group 156
Access to a Novel Class of Tetracyclic 1,4-Benzodiazepin-5-ones Starting from alpha-Aminoacids by Pd-Catalyzed Amination/1,3-Dipolar Cycloaddition as Key Steps 155
Oxidative cleavage of the isoxazolidine ring 154
Iodoamination of Alkenyl Sulfonamides by Potassium Iodide and Hydrogen Peroxide in Aqueous Medium 153
Palladium-mediated Approach to Dibenzo[b,e][1,4]diazepines and Benzopyrido-analogues. An Efficient Synthesis of Tarpane 152
Synthesis of pyrazolo[1,5-a]quinoxalines 152
A facile synthesis of 2-methyl-1,4-benzodiazepin-5-ones via intramolecular azide cycloaddition 152
Nitrilimine cycloadditions in aqueous media 151
Intramolecular nitrile imide cycloadditions onto the furan ring: synthesis of the new 3a,4-dihydro-6H-difuro[3,2-c;3,4-d]pyrazole skeleton 151
Transition metal catalyzed azidation reactions 151
Relative and absolute stereocontrol in intramolecular nitrone cycloadditions to the cyclohexene ring 150
Synthesis and Biological Evaluation of Migrastatin Macrotriazoles 149
Intramolecular Azide Cycloaddition en Route to the New Pyrrolo[2,1-c][1,2,3]triazolo[1,5-a][1,4]benzodiazepine Skeleton 148
Asymmetric induction by the (S)-1-phenylethyl group in intramolecular nitrile imine cycloadditions giving enantiopure 3,3a-dihydro-pyrazolo[1,5-alpha][1,4]benzodiazepine-4(6H)-ones 147
Efficient Synthesis of N-Methoxyindoles via Alkylative Cycloaddition of Nitrosoarenes with Alkynes 146
Entry to nitrogen-containing heterocycles by base-promoted heterocyclization on allenylamides of L-a-aminoacids 146
Synthesis of enantiopure 4-amino-6-fluoro-3-(hydroxymethyl)chromanes via intramolecular nitrone cycloadditions 146
Divergent Palladium- and Platinum-Catalyzed Intramolecular Hydroamination/Hydroarylation of O-Propargyl-2-aminophenols 146
Intramolecular cycloadditions of N-alkenoyl aryl azides 145
Intramolecular cycloadditions of nitrones derived from optically active 1-alkenyl-2-imidazolecarbaldehydes: regio- and diastereoselectivity 145
Synthesis of N-(5-amino-2-pyrimidyl)-N '-[4-(p-fluorophenyl)-4-oxobutyl]piperazine, a useful intermediate to antipsychotic agents 143
Diastereoselective nitrilimine cycloaddition to the C = N bond of enantiopure 1,4-benzodiazepinones 143
Novel aspects of the silver carbonate promoted reaction of hydrazonyl chlorides with homoallylic and homopropargylic alcohols 143
Copper-Catalyzed Alkoxylation as Key Step to Convert Isatin to Oxazinoindol-2-one Derivatives 143
Acid-mediated decarboxylative C-H coupling between arenes and O-allyl carbamates 143
Totale 19.503
Categoria #
all - tutte 100.595
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 100.595


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2021/20221.335 0 316 115 34 32 46 139 56 73 198 152 174
2022/20231.883 230 89 135 186 138 412 14 272 226 53 75 53
2023/20243.001 422 400 462 598 628 188 34 57 89 28 27 68
2024/20252.165 52 39 446 47 62 112 61 127 229 142 188 660
2025/20267.381 414 689 1.460 887 648 369 1.176 394 545 397 204 198
2026/2027280 157 123 0 0 0 0 0 0 0 0 0 0
Totale 25.822