BROGGINI, GIANLUIGI
 Distribuzione geografica
Continente #
NA - Nord America 9.809
EU - Europa 5.404
AS - Asia 1.506
SA - Sud America 49
Continente sconosciuto - Info sul continente non disponibili 16
OC - Oceania 5
AF - Africa 3
Totale 16.792
Nazione #
US - Stati Uniti d'America 9.791
IT - Italia 2.508
UA - Ucraina 1.013
TR - Turchia 510
SE - Svezia 452
VN - Vietnam 330
CN - Cina 313
IE - Irlanda 291
DE - Germania 278
SG - Singapore 263
FI - Finlandia 260
GB - Regno Unito 250
RU - Federazione Russa 151
FR - Francia 59
BR - Brasile 43
JP - Giappone 38
IN - India 26
ES - Italia 22
BE - Belgio 18
CH - Svizzera 17
EU - Europa 16
CA - Canada 15
CZ - Repubblica Ceca 15
NL - Olanda 15
AT - Austria 13
PT - Portogallo 8
RO - Romania 7
NO - Norvegia 6
AU - Australia 5
BD - Bangladesh 4
BG - Bulgaria 4
DK - Danimarca 3
GR - Grecia 3
ID - Indonesia 3
IL - Israele 3
IQ - Iraq 3
PL - Polonia 3
AZ - Azerbaigian 2
BO - Bolivia 2
MY - Malesia 2
PA - Panama 2
UY - Uruguay 2
AE - Emirati Arabi Uniti 1
AL - Albania 1
BN - Brunei Darussalam 1
BT - Bhutan 1
BY - Bielorussia 1
DZ - Algeria 1
EC - Ecuador 1
EG - Egitto 1
ET - Etiopia 1
HU - Ungheria 1
JO - Giordania 1
KZ - Kazakistan 1
LU - Lussemburgo 1
MD - Moldavia 1
ME - Montenegro 1
MM - Myanmar 1
MO - Macao, regione amministrativa speciale della Cina 1
MX - Messico 1
SI - Slovenia 1
SK - Slovacchia (Repubblica Slovacca) 1
TH - Thailandia 1
TW - Taiwan 1
VE - Venezuela 1
Totale 16.792
Città #
Milan 1.728
Fairfield 1.649
Woodbridge 927
Jacksonville 780
Ashburn 768
Houston 667
Seattle 659
Chandler 628
Wilmington 560
Cambridge 506
Ann Arbor 391
Dearborn 378
Dublin 291
Princeton 280
Nyköping 279
Izmir 224
Dong Ket 211
Boardman 187
Singapore 136
Rome 130
San Mateo 109
San Diego 97
Como 73
Chicago 66
Ogden 55
Kocaeli 50
Beijing 46
London 42
Santa Clara 39
Tokyo 36
Kunming 33
Washington 32
Düsseldorf 31
Hefei 31
Verona 28
Dallas 18
Los Angeles 18
Nanjing 18
Nanchang 17
New York 16
Norwalk 16
Brussels 15
Munich 15
Brno 13
Clausthal-Zellerfeld 13
Berlin 12
Fuzhou 12
Helsinki 12
Jinan 12
West Jordan 12
Guangzhou 11
Kilburn 11
Toronto 11
Vienna 11
Frankfurt am Main 10
Bari 9
Chiswick 9
Hounslow 9
Paris 9
Rotonda 9
Auburn Hills 8
Council Bluffs 8
Edinburgh 8
New Bedfont 8
Nuremberg 8
Shanghai 8
Lappeenranta 7
North Bergen 7
Prescot 7
São Paulo 7
Cavaria con Premezzo 6
Florence 6
Islington 6
Lisbon 6
New Delhi 6
Oslo 6
Timisoara 6
Acton 5
Amsterdam 5
Besana In Brianza 5
Brescia 5
Changsha 5
Giussano 5
Perugia 5
Philadelphia 5
Phoenix 5
Rozzano 5
San Francisco 5
Shenyang 5
Southwark 5
Wandsworth 5
Wuhan 5
Bristol 4
Chengdu 4
Hebei 4
Madrid 4
Mumbai 4
Naples 4
Redmond 4
Rouen 4
Totale 12.690
Nome #
1,3-Dipolar cycloadditions to nitrogen-substituted allenes 282
1,3-Dipolar cycloadditions to allenes 208
C-C, C-O, C-N Bond Formation on sp2-Carbon by Pd(II)-Catalyzed Reactions Involving Oxidant Agents 191
Boehmeriasin A as new lead compound for the inhibition of topoisomerases and SIRT2 190
Copper(II)-catalyzed alkoxyhalogenation of alkynyl ureas and amides as a route to haloalkylidene substituted heterocycles 177
Palladium-catalyzed domino carbopalladation/5-exo-allylic amination of α-amino allenamides: an efficient entry to enantiopure imidazolidinones 174
Synthesis and biological evaluation of 1,7,8,8a-tetrahydro-3H-oxazolo[3,4-a]pyrazin-6(5H)-ones as antitumoral agents 173
Stereoselective intramolecular cycloadditions of homochiral nitrile imines: synthesis of enantiomerically pure 3,3a-dihydro-pyrazolo[1,5-a][1,4] benzodiazepine-6(4H)-ones 172
Synthesis of Pironetin-Dumetorine Hybrids as Tubulin Binders 168
(Diacyloxyiodo)benzenes-Driven Palladium-Catalyzed Cyclizations of Unsaturated N-Sulfonylamides: Opportunities of Path Selection 167
A facile synthesis of flumazenil analogues 166
An alternative synthesis of 2-alkylidene-3,4-dihydro-2H-1,4-benzoxazines by intramolecular gold-catalyzed hydroalkoxylation of 2-(prop-2-yn-1-ylamino)-phenols 163
Selective intramolecular palladium(II)-catalyzed aminooxygenation vs. diamination of alkenylureas: efficient microwave-assisted reactions to bicyclic piperazinones 162
SYNTHESIS OF ENANTIOPURE 4-AMINO-3-HYDROXYMETHYL-TETRAHYDROQUINOLINES VIA AN INTRAMOLECULAR NITRONE CYCLOADDITION 160
Intramolecular Oxidative Palladium-Catalyzed Amination Involving Double C-H Functionalization of Unactivated Olefins 160
A synthetic route to [1,2,4]triazolo[1,5-a][4,1]benzoxazepines 156
Solvent- and ligand-free palladium-catalyzed amination of aryl halides 156
A New Entry to [1,2,4]Triazolo[1,5-a][1,4]benzodiazepin-6-ones via Intramolecular Nitrilimine Cycloaddition to the Cyano Group 154
Ruthenium-Catalyzed Hydroamination of Aminoallenes: an Approach to Vinyl Substituted Heterocycles 154
Synthesis of 1,4-benzodiazepinones via palladium-catalysed allene carbopalladation/amination domino sequence 154
Intra-Intermolecular Palladium-Catalyzed Domino Reactions of Glycine Allylamides for the Synthesis of Diversely Functionalized Piperazinones 153
New Mechanistic Evidence on the Reaction between Sulfonylallenes and Nitrile Oxides 151
Palladium(II)/copper halide/solvent combination for selective intramolecular domino reactions of indole carboxylic acid allylamides. An unprecedented arylation/esterification sequence 149
Transition metal complexation in 1,3-dipolar cycloadditions 149
Access to pyrrolo-pyridines by gold-catalyzed hydroarylation of pyrroles tethered to terminal alkynes 146
Dehydrogenative Allylic Aminations of But-3-enoic Acid Derivatives 146
The intramolecular azide cycloaddition route to triazolam analogues 146
Intramolecular azide cycloadditions leading to [1,2,3]triazolo[1,5-a]quinoxalines 146
Diastereoselective synthesis of bis(3,5)pyrazolophanes by sequential inter- and intramolecular cycloadditions of homochiral nitrilimines 142
New Access to Kainic Acid via Intramolecular Palladium-Catalyzed Allylic Alkylation 141
Palladium-Catalyzed Cyclization/Carbonylation as a Direct Route to 4-[(Methoxycarbonyl)methyl]-3,4-dihydroisoquinolinones 140
Recent advances in heterobimetallic palladium(ii)/copper(ii) catalyzed domino difunctionalization of carbon–carbon multiple bonds 140
N,N-Disubstituted Propargylamines as Tools in the Sequential 1,3-Dipolar Cycloaddition/Arylation Processes to the Formation of Polyheterocyclic Systems 140
Synthesis of Bis-(3,5)pyrazolophanes by Sequential Intermolecular-Intramolecular Nitrilimine Cycloadditions 139
Synthesis of enantiopure 3-hydroxymethylchromanes via intramolecular nitrone cycloaddition 139
Palladium-Catalysed Carbo- and Hydroamination of Allenyl Ethers and Aminoallenes: Available Entry to Nitrogen-Containing Benzo-Fused Rings 139
5-Heterosubstituted 4-methylene-4,5-dihydroisoxazoles: Ready accessibility and versatile reactivity 137
Thermal behaviour of dipolarophile-containing acyl azides: intramolecular cycloaddition versus Curtius rearrangement 136
Intramolecular oxidative palladium-catalyzed diamination reactions of alkenyl sulfamates: an efficient synthesis of [1,2,5]thiadiazolo-fused piperazinones 136
The first case of asymmetric induction in intramolecular nitrile imine cycloadditions: synthesis of enantiopure 3-substituted 6-oxo-2,3,3a,5-tetrahydro-4-carbomethoxy-furo[3,4-c]pyrazoles 134
Efficient Approach to the Unknown Isoxazolo[3,4-d]thieno[2,3-b]pyridine System by Regioselective Intramolecular Nitrone Cycloadditions 134
Synthetic approach to imidazo[1,2-a]pyridine derivatives by the intramolecular nitrone cycloaddition methodology 133
Regiochemical aspects of intramolecular cycloadditions of nitrones derived from N-(2-alkenyl)-2-pyrrolecarbaldehydes. Competitive entries to pyrrolizidine and indolizidine derivatives 133
Solvent-free, microwave-assisted N-arylation of indolines by using low palladium catalyst loadings 133
Transition metal-catalyzed hydroamination and carboamination reactions of anthranilic allenamides as a route to 2-vinyl- and 2-(a-styryl)-quinazolin-4-one derivatives 133
Intramolecular Cycloadditions of Nitrones Derived from 1-Allyl-2-pyrrolecarbaldehyde as a Route to Racemic and Enantiopure Pyrrolizidines and Indolizidines 132
Uncommon intramolecular palladium-catalyzed cyclization of indole derivatives 132
Dipolarophilic behavior of the isoxazole ring in intramolecular nitrilimine cycloadditions 132
Pyrrolizidine and indolizidine syntheses involving 1,3-dipolar cycloadditions 132
A valuable approach to enantiopure partially saturated pyrrolo- and indolo[1,2-a]indoles by intramolecular nitrone cycloadditions to the cyclohexene ring 131
Dipolarophilic behaviour of (arylsulfonyl)allenes towards nitrilimines 131
Intramolecular Palladium-Catalyzed Aminocarboxylation of Olefins as a Direct Route to Bicyclic Oxazolidinones 131
Palladium-Catalyzed dual C-H or N-H functionalization of unfunctionalized indole derivatives with alkenes and arenes 131
Intramolecular oxidative Pd(II)-catalyzed alkoxylation of 3-aza-5-alkenols with O2 as sole oxidant: mild conditions for the synthesis of 1,4-oxazine derivatives 130
Stereoselective intramolecular cycloadditions of homochiral N-alkenoyl aryl azides 129
L-alanine benzylester as chiral inductor: Synthesis of enantiopure pyrazolo[1,5-a]-[1,4]benzodiazepine-4-ones via intramolecular nitrilimine cycloadditions 128
Regioselective Intramolecular Cycloaddition of C-(1-Acryloyl-2-pyrrolyl)-N-benzylnitrone: Entry to 6-Hydroxy-5-oxoindolizidines 127
Palladium-mediated Approach to Dibenzo[b,e][1,4]diazepines and Benzopyrido-analogues. An Efficient Synthesis of Tarpane 127
Intramolecular Pd(II)-Catalyzed Cyclization of Propargylamides: Straightforward Synthesis of 5-Oxazole-carbaldehydes 127
Pd-Catalyzed Intramolecular Cyclization of Pyrrolo-2-carboxamides: Regiodivergent Routes to Pyrrolo-pyrazines and Pyrrolo-pyridines 126
Palladium-catalyzed C-N bond formation via direct C-H bond functionalization. Recent developments in heterocyclic synthesis 126
Enantiopure 2-piperidylacetaldehyde as useful building block in the diversity-oriented synthesis of polycyclic piperidine derivatives 126
Synthesis of tetrazolo[1,5-a][1,4]benzodiazepin-6-ones via intramolecular azide cycloadditions onto the cyano group 126
A valuable heterocyclic ring transformation: from isoxazolin-5(2H)-ones to quinolines 125
Regioselectivity on the palladium-catalyzed intramolecular cyclization of indole derivatives 124
Synthesis of enantiopure pyrrolo[3,4-c]pyrazole derivatives via intramolecular cycloaddition of homochiral nitrilimines 123
Synthesis of enantiopure 4-amino-6-fluoro-3-(hydroxymethyl)chromanes via intramolecular nitrone cycloadditions 123
A new protocol for the conversion of isoxazolidines to 1,3-aminoalcohols 120
Synthesis and Biological Evaluation of Migrastatin Macrotriazoles 120
Intramolecular cycloadditions of N-alkenoyl aryl azides 119
Diastereoselective nitrilimine cycloaddition to the C = N bond of enantiopure 1,4-benzodiazepinones 119
Nitrilimine cycloadditions onto partially saturated furo[3,4-c]thieno[2,3-d]pyrazoles. A problem in site selectivity 119
Relative and absolute stereocontrol in intramolecular nitrone cycloadditions to the cyclohexene ring 119
Divergent Palladium- and Platinum-Catalyzed Intramolecular Hydroamination/Hydroarylation of O-Propargyl-2-aminophenols 119
Intramolecular Aminoazidation of Unactivated Terminal Alkenes by Palladium-Catalyzed Reactions with Hydrogen Peroxide as the Oxidant 119
Intramolecular Azide Cycloaddition en Route to the New Pyrrolo[2,1-c][1,2,3]triazolo[1,5-a][1,4]benzodiazepine Skeleton 118
Intramolecular nitrile imide cycloadditions onto the furan ring: synthesis of the new 3a,4-dihydro-6H-difuro[3,2-c;3,4-d]pyrazole skeleton 117
Efficient Synthesis of N-Methoxyindoles via Alkylative Cycloaddition of Nitrosoarenes with Alkynes 116
Synthesis of pyrazolo[1,5-a]quinoxalines 116
Nitrilimine cycloadditions in aqueous media 114
A new synthesis of flumazenil suitable for fluorine-18 labeling 114
Intramolecular cycloadditions of nitrones derived from optically active 1-alkenyl-2-imidazolecarbaldehydes: regio- and diastereoselectivity 114
Microwave-Assisted Intramolecular Cyclization of Electron-Rich HeterocycleDerivatives by a Palladium-Catalyzed Coupling Reaction 114
Copper-Catalyzed Alkoxylation as Key Step to Convert Isatin to Oxazinoindol-2-one Derivatives 114
Synthesis of 5-hydroxymethyl-1,4-dioxan-2-one 113
Tunable Pd-Catalyzed Cyclization of Indole-2-carboxylic Acid Allenamides: Carboamination vs Microwave-Assisted Hydroamination 113
Selective 7- endo -Cyclization of 3-Aza-5-alkenols through Oxidative Pd(II)-Catalyzed Olefin Oxyarylation 113
Chimica degli eterocicli 112
Enantioselective intramolecular nitrone cycloaddition route to 3-(trifluoromethyl)-isoxazolidino[4,3-c]-chroman-4-ones and -quinolin-4-ones 112
Dipolarophilic behaviour of the thiophene ring in intramolecular nitrile imine cycloadditions 110
Novel aspects of the silver carbonate promoted reaction of hydrazonyl chlorides with homoallylic and homopropargylic alcohols 110
A Valuable Synthesis of Pyrrolo[1,2-a]quinoxalines, Indolo[1,2-a]quinoxalines and their Aza-Analogues by Palladium-Catalyzed Intramolecular Carbon-Nitrogen Bond Formation 109
Oxidative cleavage of the isoxazolidine ring 109
Synthesis of N-(5-amino-2-pyrimidyl)-N '-[4-(p-fluorophenyl)-4-oxobutyl]piperazine, a useful intermediate to antipsychotic agents 107
Effective Synthesis of Enantiopure [1,2,3]Triazolo[1,5-a]- and Pyrazolo[1,5-a]-pyrrolo[2,1-c][1,4]benzodiazepines by Diastereoselective Intramolecular Azide and Nitrilimine Cycloadditions 107
Synthesis and biological evaluation of pyrimidine-oxazolidin-2-arylimino hybrid molecules as antibacterial agents 107
Pd-Catalyzed Cyclization of 1-Allyl-2-indolecarboxamides by Intramolecular Amidation of Unactivated Ethylenic Bond 105
Access to pyrralo- and pyrido[1,2-a]indole derivatives by intramolecular nitrone cycloadditions. Effect of steric factors on the regioselective product formation 104
Site-selective and regioselective cycloaddition of N-propadienylanilines with nitrile oxides. Claisen-type rearrangement of the cycloadducts 103
Synthesis of pyrazole-containing azacrown ethers by intramolecular nitrilimine cycloadditions 102
Totale 13.548
Categoria #
all - tutte 71.363
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 71.363


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2019/2020798 0 0 0 0 0 0 0 0 281 242 62 213
2020/20212.423 56 233 106 228 130 262 162 203 330 181 203 329
2021/20221.507 172 316 115 34 32 46 139 56 73 198 152 174
2022/20231.883 230 89 135 186 138 412 14 272 226 53 75 53
2023/20243.001 422 400 462 598 628 188 34 57 89 28 27 68
2024/20251.040 52 39 446 47 62 112 61 127 94 0 0 0
Totale 17.036