BROGGINI, GIANLUIGI
 Distribuzione geografica
Continente #
NA - Nord America 15.997
EU - Europa 6.200
AS - Asia 4.282
SA - Sud America 453
Continente sconosciuto - Info sul continente non disponibili 266
AF - Africa 74
OC - Oceania 6
Totale 27.278
Nazione #
US - Stati Uniti d'America 15.759
IT - Italia 2.740
SG - Singapore 1.380
UA - Ucraina 1.021
CN - Cina 940
VN - Vietnam 638
TR - Turchia 523
SE - Svezia 516
HK - Hong Kong 458
BR - Brasile 376
GB - Regno Unito 367
DE - Germania 352
FI - Finlandia 297
IE - Irlanda 293
FR - Francia 206
RU - Federazione Russa 173
CA - Canada 115
IN - India 101
JP - Giappone 72
MX - Messico 71
ES - Italia 52
BD - Bangladesh 42
PL - Polonia 33
ZA - Sudafrica 31
IQ - Iraq 27
NL - Olanda 25
AR - Argentina 24
BE - Belgio 19
CH - Svizzera 18
EU - Europa 16
CZ - Repubblica Ceca 15
NG - Nigeria 15
AT - Austria 13
VE - Venezuela 13
ID - Indonesia 12
AE - Emirati Arabi Uniti 10
EC - Ecuador 9
LT - Lituania 9
PK - Pakistan 9
PT - Portogallo 8
SA - Arabia Saudita 8
JM - Giamaica 7
MD - Moldavia 7
RO - Romania 7
TN - Tunisia 7
AU - Australia 6
CL - Cile 6
CO - Colombia 6
IL - Israele 6
NO - Norvegia 6
NP - Nepal 6
PE - Perù 6
GT - Guatemala 5
HN - Honduras 5
MY - Malesia 5
PH - Filippine 5
PY - Paraguay 5
TT - Trinidad e Tobago 5
UZ - Uzbekistan 5
AZ - Azerbaigian 4
BB - Barbados 4
BG - Bulgaria 4
GR - Grecia 4
JO - Giordania 4
KE - Kenya 4
SV - El Salvador 4
TH - Thailandia 4
TW - Taiwan 4
UY - Uruguay 4
BO - Bolivia 3
CR - Costa Rica 3
DK - Danimarca 3
EG - Egitto 3
GP - Guadalupe 3
KZ - Kazakistan 3
MA - Marocco 3
NI - Nicaragua 3
PA - Panama 3
PR - Porto Rico 3
ZW - Zimbabwe 3
AL - Albania 2
BN - Brunei Darussalam 2
DM - Dominica 2
DZ - Algeria 2
HU - Ungheria 2
LB - Libano 2
OM - Oman 2
PS - Palestinian Territory 2
SN - Senegal 2
BH - Bahrain 1
BS - Bahamas 1
BT - Bhutan 1
BY - Bielorussia 1
CI - Costa d'Avorio 1
DO - Repubblica Dominicana 1
EE - Estonia 1
ET - Etiopia 1
GA - Gabon 1
GD - Grenada 1
GY - Guiana 1
Totale 27.013
Città #
Dallas 1.920
Milan 1.770
Fairfield 1.650
Ashburn 1.320
San Jose 1.093
Woodbridge 927
Singapore 812
Jacksonville 784
Houston 690
Seattle 671
Chandler 628
Wilmington 563
Cambridge 506
Hong Kong 451
Council Bluffs 446
Ann Arbor 391
Dearborn 380
Dublin 293
Princeton 280
Nyköping 279
Izmir 224
Dong Ket 211
Beijing 200
The Dalles 196
Boardman 189
Chicago 164
Rome 149
Los Angeles 139
Lauterbourg 127
Washington 117
San Mateo 109
Santa Clara 108
Ho Chi Minh City 105
San Diego 101
New York 94
Como 76
Hanoi 76
London 74
Tokyo 66
Munich 63
São Paulo 62
Orem 58
Ogden 55
Kocaeli 50
Mexico City 45
Atlanta 34
Guangzhou 34
Montreal 34
Phoenix 34
Kunming 33
Buffalo 32
Des Moines 32
Düsseldorf 32
Hefei 32
Turku 32
Chennai 31
Verona 30
Manchester 28
Shanghai 28
Brooklyn 27
Warsaw 27
Toronto 25
Denver 24
Johannesburg 24
Boston 22
Mumbai 21
Stockholm 21
Varese 21
Nanjing 19
Naples 19
Frankfurt am Main 18
Nanchang 18
San Francisco 18
Hangzhou 17
Helsinki 17
Norwalk 17
Paris 17
Philadelphia 17
Brussels 16
Las Vegas 16
Abuja 15
Da Nang 15
Amsterdam 14
Bari 14
North Bergen 14
Brno 13
Clausthal-Zellerfeld 13
Fuzhou 13
Jinan 13
Nuremberg 13
Shenzhen 13
Berlin 12
Elk Grove Village 12
Poplar 12
Rio de Janeiro 12
West Jordan 12
Kilburn 11
Vienna 11
Baghdad 10
Campinas 10
Totale 19.831
Nome #
1,3-Dipolar cycloadditions to nitrogen-substituted allenes 1.215
1,3-Dipolar cycloadditions to allenes 1.211
C-C, C-O, C-N Bond Formation on sp2-Carbon by Pd(II)-Catalyzed Reactions Involving Oxidant Agents 284
Palladium-catalyzed domino carbopalladation/5-exo-allylic amination of α-amino allenamides: an efficient entry to enantiopure imidazolidinones 282
Boehmeriasin A as new lead compound for the inhibition of topoisomerases and SIRT2 268
Dipolarophilic behavior of the isoxazole ring in intramolecular nitrilimine cycloadditions 247
A facile synthesis of flumazenil analogues 237
Copper(II)-catalyzed alkoxyhalogenation of alkynyl ureas and amides as a route to haloalkylidene substituted heterocycles 234
Synthesis and biological evaluation of 1,7,8,8a-tetrahydro-3H-oxazolo[3,4-a]pyrazin-6(5H)-ones as antitumoral agents 229
(Diacyloxyiodo)benzenes-Driven Palladium-Catalyzed Cyclizations of Unsaturated N-Sulfonylamides: Opportunities of Path Selection 229
A synthetic route to [1,2,4]triazolo[1,5-a][4,1]benzoxazepines 228
Synthesis of Pironetin-Dumetorine Hybrids as Tubulin Binders 227
An alternative synthesis of 2-alkylidene-3,4-dihydro-2H-1,4-benzoxazines by intramolecular gold-catalyzed hydroalkoxylation of 2-(prop-2-yn-1-ylamino)-phenols 221
Intramolecular Oxidative Palladium-Catalyzed Amination Involving Double C-H Functionalization of Unactivated Olefins 221
Stereoselective intramolecular cycloadditions of homochiral nitrile imines: synthesis of enantiomerically pure 3,3a-dihydro-pyrazolo[1,5-a][1,4] benzodiazepine-6(4H)-ones 221
A New Entry to [1,2,4]Triazolo[1,5-a][1,4]benzodiazepin-6-ones via Intramolecular Nitrilimine Cycloaddition to the Cyano Group 219
Synthesis of 1,4-benzodiazepinones via palladium-catalysed allene carbopalladation/amination domino sequence 210
A valuable approach to enantiopure partially saturated pyrrolo- and indolo[1,2-a]indoles by intramolecular nitrone cycloadditions to the cyclohexene ring 209
Ruthenium-Catalyzed Hydroamination of Aminoallenes: an Approach to Vinyl Substituted Heterocycles 207
Access to pyrrolo-pyridines by gold-catalyzed hydroarylation of pyrroles tethered to terminal alkynes 206
Intra-Intermolecular Palladium-Catalyzed Domino Reactions of Glycine Allylamides for the Synthesis of Diversely Functionalized Piperazinones 204
Selective intramolecular palladium(II)-catalyzed aminooxygenation vs. diamination of alkenylureas: efficient microwave-assisted reactions to bicyclic piperazinones 202
SYNTHESIS OF ENANTIOPURE 4-AMINO-3-HYDROXYMETHYL-TETRAHYDROQUINOLINES VIA AN INTRAMOLECULAR NITRONE CYCLOADDITION 198
Palladium-Catalysed Carbo- and Hydroamination of Allenyl Ethers and Aminoallenes: Available Entry to Nitrogen-Containing Benzo-Fused Rings 198
Palladium(II)/copper halide/solvent combination for selective intramolecular domino reactions of indole carboxylic acid allylamides. An unprecedented arylation/esterification sequence 197
5-Heterosubstituted 4-methylene-4,5-dihydroisoxazoles: Ready accessibility and versatile reactivity 197
Recent advances in heterobimetallic palladium(ii)/copper(ii) catalyzed domino difunctionalization of carbon–carbon multiple bonds 194
Intramolecular oxidative palladium-catalyzed diamination reactions of alkenyl sulfamates: an efficient synthesis of [1,2,5]thiadiazolo-fused piperazinones 194
Solvent- and ligand-free palladium-catalyzed amination of aryl halides 192
Diastereoselective synthesis of bis(3,5)pyrazolophanes by sequential inter- and intramolecular cycloadditions of homochiral nitrilimines 190
Efficient Approach to the Unknown Isoxazolo[3,4-d]thieno[2,3-b]pyridine System by Regioselective Intramolecular Nitrone Cycloadditions 190
New Mechanistic Evidence on the Reaction between Sulfonylallenes and Nitrile Oxides 188
Synthesis of enantiopure 3-hydroxymethylchromanes via intramolecular nitrone cycloaddition 188
The intramolecular azide cycloaddition route to triazolam analogues 188
A valuable heterocyclic ring transformation: from isoxazolin-5(2H)-ones to quinolines 186
Transition metal complexation in 1,3-dipolar cycloadditions 184
Palladium-Catalyzed dual C-H or N-H functionalization of unfunctionalized indole derivatives with alkenes and arenes 183
Regioselective Intramolecular Cycloaddition of C-(1-Acryloyl-2-pyrrolyl)-N-benzylnitrone: Entry to 6-Hydroxy-5-oxoindolizidines 182
A new synthesis of flumazenil suitable for fluorine-18 labeling 182
Intramolecular oxidative Pd(II)-catalyzed alkoxylation of 3-aza-5-alkenols with O2 as sole oxidant: mild conditions for the synthesis of 1,4-oxazine derivatives 182
Intramolecular azide cycloadditions leading to [1,2,3]triazolo[1,5-a]quinoxalines 182
Pyrrolizidine and indolizidine syntheses involving 1,3-dipolar cycloadditions 181
Palladium-catalyzed C-N bond formation via direct C-H bond functionalization. Recent developments in heterocyclic synthesis 181
Dehydrogenative Allylic Aminations of But-3-enoic Acid Derivatives 181
N,N-Disubstituted Propargylamines as Tools in the Sequential 1,3-Dipolar Cycloaddition/Arylation Processes to the Formation of Polyheterocyclic Systems 181
Synthesis of Bis-(3,5)pyrazolophanes by Sequential Intermolecular-Intramolecular Nitrilimine Cycloadditions 180
New Access to Kainic Acid via Intramolecular Palladium-Catalyzed Allylic Alkylation 178
Intramolecular Pd(II)-Catalyzed Cyclization of Propargylamides: Straightforward Synthesis of 5-Oxazole-carbaldehydes 178
Transition metal-catalyzed hydroamination and carboamination reactions of anthranilic allenamides as a route to 2-vinyl- and 2-(a-styryl)-quinazolin-4-one derivatives 178
Intramolecular Aminoazidation of Unactivated Terminal Alkenes by Palladium-Catalyzed Reactions with Hydrogen Peroxide as the Oxidant 177
Chimica degli eterocicli 176
Enantiopure 2-piperidylacetaldehyde as useful building block in the diversity-oriented synthesis of polycyclic piperidine derivatives 176
Thermal behaviour of dipolarophile-containing acyl azides: intramolecular cycloaddition versus Curtius rearrangement 176
Intramolecular Cycloadditions of Nitrones Derived from 1-Allyl-2-pyrrolecarbaldehyde as a Route to Racemic and Enantiopure Pyrrolizidines and Indolizidines 174
Uncommon intramolecular palladium-catalyzed cyclization of indole derivatives 174
The first case of asymmetric induction in intramolecular nitrile imine cycloadditions: synthesis of enantiopure 3-substituted 6-oxo-2,3,3a,5-tetrahydro-4-carbomethoxy-furo[3,4-c]pyrazoles 174
L-alanine benzylester as chiral inductor: Synthesis of enantiopure pyrazolo[1,5-a]-[1,4]benzodiazepine-4-ones via intramolecular nitrilimine cycloadditions 174
Regiochemical aspects of intramolecular cycloadditions of nitrones derived from N-(2-alkenyl)-2-pyrrolecarbaldehydes. Competitive entries to pyrrolizidine and indolizidine derivatives 173
Palladium-mediated Approach to Dibenzo[b,e][1,4]diazepines and Benzopyrido-analogues. An Efficient Synthesis of Tarpane 171
A Valuable Synthesis of Pyrrolo[1,2-a]quinoxalines, Indolo[1,2-a]quinoxalines and their Aza-Analogues by Palladium-Catalyzed Intramolecular Carbon-Nitrogen Bond Formation 171
Palladium-Catalyzed Cyclization/Carbonylation as a Direct Route to 4-[(Methoxycarbonyl)methyl]-3,4-dihydroisoquinolinones 171
Solvent-free, microwave-assisted N-arylation of indolines by using low palladium catalyst loadings 171
A new protocol for the conversion of isoxazolidines to 1,3-aminoalcohols 171
Intramolecular nitrile imide cycloadditions as a synthetic strategy to macrocyclic heterophanes containing pyrazole unit(s) 171
Synthesis of tetrazolo[1,5-a][1,4]benzodiazepin-6-ones via intramolecular azide cycloadditions onto the cyano group 171
Pd-Catalyzed Intramolecular Cyclization of Pyrrolo-2-carboxamides: Regiodivergent Routes to Pyrrolo-pyrazines and Pyrrolo-pyridines 170
Enantioselective intramolecular nitrone cycloaddition route to 3-(trifluoromethyl)-isoxazolidino[4,3-c]-chroman-4-ones and -quinolin-4-ones 170
Synthetic approach to imidazo[1,2-a]pyridine derivatives by the intramolecular nitrone cycloaddition methodology 169
Stereoselective intramolecular cycloadditions of homochiral N-alkenoyl aryl azides 168
Synthesis of enantiopure pyrrolo[3,4-c]pyrazole derivatives via intramolecular cycloaddition of homochiral nitrilimines 168
Intramolecular Palladium-Catalyzed Aminocarboxylation of Olefins as a Direct Route to Bicyclic Oxazolidinones 167
Nitrilimine cycloadditions onto partially saturated furo[3,4-c]thieno[2,3-d]pyrazoles. A problem in site selectivity 166
Dipolarophilic behaviour of (arylsulfonyl)allenes towards nitrilimines 165
Dipolarophilic behaviour of the thiophene ring in intramolecular nitrile imine cycloadditions 165
Selective 7- endo -Cyclization of 3-Aza-5-alkenols through Oxidative Pd(II)-Catalyzed Olefin Oxyarylation 165
Direct Synthesis of Fluorescent Oxazolo-phenoxazines by Copper-Catalyzed/Hypervalent Iodine(III)-Mediated Dimerization/Cyclization of 2-Benzylamino-phenols 165
Access to pyrralo- and pyrido[1,2-a]indole derivatives by intramolecular nitrone cycloadditions. Effect of steric factors on the regioselective product formation 164
Regioselectivity on the palladium-catalyzed intramolecular cyclization of indole derivatives 163
Synthesis of pyrazolo[1,5-a]quinoxalines 163
Access to a Novel Class of Tetracyclic 1,4-Benzodiazepin-5-ones Starting from alpha-Aminoacids by Pd-Catalyzed Amination/1,3-Dipolar Cycloaddition as Key Steps 162
Intramolecular nitrile imide cycloadditions onto the furan ring: synthesis of the new 3a,4-dihydro-6H-difuro[3,2-c;3,4-d]pyrazole skeleton 162
Oxidative cleavage of the isoxazolidine ring 161
A facile synthesis of 2-methyl-1,4-benzodiazepin-5-ones via intramolecular azide cycloaddition 161
Iodoamination of Alkenyl Sulfonamides by Potassium Iodide and Hydrogen Peroxide in Aqueous Medium 160
Nitrilimine cycloadditions in aqueous media 159
Synthesis and Biological Evaluation of Migrastatin Macrotriazoles 157
Transition metal catalyzed azidation reactions 157
Synthesis of enantiopure 4-amino-6-fluoro-3-(hydroxymethyl)chromanes via intramolecular nitrone cycloadditions 155
Relative and absolute stereocontrol in intramolecular nitrone cycloadditions to the cyclohexene ring 155
Asymmetric induction by the (S)-1-phenylethyl group in intramolecular nitrile imine cycloadditions giving enantiopure 3,3a-dihydro-pyrazolo[1,5-alpha][1,4]benzodiazepine-4(6H)-ones 153
Efficient Synthesis of N-Methoxyindoles via Alkylative Cycloaddition of Nitrosoarenes with Alkynes 153
Intramolecular Azide Cycloaddition en Route to the New Pyrrolo[2,1-c][1,2,3]triazolo[1,5-a][1,4]benzodiazepine Skeleton 152
Copper-Catalyzed Alkoxylation as Key Step to Convert Isatin to Oxazinoindol-2-one Derivatives 152
Divergent Palladium- and Platinum-Catalyzed Intramolecular Hydroamination/Hydroarylation of O-Propargyl-2-aminophenols 152
Synthesis of N-(5-amino-2-pyrimidyl)-N '-[4-(p-fluorophenyl)-4-oxobutyl]piperazine, a useful intermediate to antipsychotic agents 151
Intramolecular cycloadditions of nitrones derived from optically active 1-alkenyl-2-imidazolecarbaldehydes: regio- and diastereoselectivity 150
Entry to nitrogen-containing heterocycles by base-promoted heterocyclization on allenylamides of L-a-aminoacids 150
Construction of the pyrazolo [1,5-a][4,1]benzothiazepine system by intramolecular nitrile imine cycloaddition 150
Synthesis of 5-hydroxymethyl-1,4-dioxan-2-one 150
Intramolecular cycloadditions of N-alkenoyl aryl azides 149
Totale 20.394
Categoria #
all - tutte 106.602
article - articoli 0
book - libri 0
conference - conferenze 0
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 106.602


Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2021/2022904 0 0 0 34 32 46 139 56 73 198 152 174
2022/20231.883 230 89 135 186 138 412 14 272 226 53 75 53
2023/20243.001 422 400 462 598 628 188 34 57 89 28 27 68
2024/20252.165 52 39 446 47 62 112 61 127 229 142 188 660
2025/20267.381 414 689 1.460 887 648 369 1.176 394 545 397 204 198
2026/20271.736 157 331 724 524 0 0 0 0 0 0 0 0
Totale 27.278